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Adrenergic Receptor Antagonist/Agonists

Other Endocrinology & Hormones Related Inhibitors

Androgen Receptor Estrogen/progestogen Receptor Aromatase 5-alpha Reductase RAAS Glucocorticoid Receptor ACE Mineralocorticoid Receptor PGDS Progesterone Receptor

Isoform-selective Products

Cat.No. Product Name Information Product Use Citations Product Validations
S4009 Mirabegron Mirabegron (YM 178) is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.
Frontiers in Pharmacology, October 25, 2022, 1008085
Biomed Pharmacother, 2025, 183:117816
iScience, 2024, 27(10):110862
S4076 Propranolol HCl Propranolol HCl (AY-64043, ICI-45520, NCS-91523) is a competitive non-selective beta-adrenergic receptors inhibitor.
Frontiers in Endocrinology, June 23, 2022, 895360
Oncology Reports, July 23, 2021, 202
Investigative Ophthalmology & Visual Science, February 2, 2026, 15
S2521 Epinephrine bitartrate Epinephrine bitartrate (Adrenalinium) is an alpha- and beta-adrenergic receptor stimulator.
Science Advances, August 16, 2024, eado1533
International Journal of Biological Sciences, April 2, 2023, 2006-2019
Advanced Science, 2025, e13580
S9507 (−)-Norepinephrine (−)-Norepinephrine (Arterenol, Levarterenol, L-Noradrenaline) is a natural neurotransmitter and hormone. It is an agonist of adrenergic receptors with Ki values of 330, 56, and 740 nM for α1, α2, and β1 adrenoceptors, respectively.This compound can be used to induce animal models of Cardiomyopathy.
ERJ Open Research, September 4, 2025, 00342-2025
ERJ Open Research, September 04, 2025, 00342-2025
Nature Communications, October 6, 2025, 8870
S2566 Isoprenaline (Isoproterenol) HCl Isoprenaline (Isoproterenol) HCl is a non-selective beta-adrenergic receptor agonist, used for the treatment of bradycardia and heart block.
Advanced Science, 2025, e00376
International Journal of Biological Sciences, 2025, 6430-6451
Animal Nutrition, 2025, 1-16
S1831 Carvedilol Carvedilol (BM-14190, SKF 105517) is a non-selective beta blocker/alpha-1 blocker, used to treat congestive heart failure (CHF) and high blood pressure.
Communications Medicine, 2025, 420
Gastroenterology, 2024, 167(5):993-1007
J Immunother Cancer, 2024, 12(11)e009805
S2516 Xylazine HCl Xylazine(BAY 1470 hydrochloride) is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant.
J Immunother Cancer, 2024, 12(11)e009805
Cell Death Dis, 2023, 14(5):318
Cell Death & Disease, 2022, 351
S2569 Phenylephrine HCl Phenylephrine HCl is a selective α1-adrenergic receptor agonist, used primarily as a decongestant.
Circulation Research, 2026, nan
J Am Heart Assoc, 2025, 14(1):e037400
NPJ Regen Med, 2023, 8(1):9
Verified customer review of Phenylephrine HCl
S8114 ICI 118551 Hydrochloride (Zenidolol) Zenidolol (ICI-118551) Hydrochloride is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
Immunity, 2025, S1074-7613(25)00226-2
Advanced Science, 2025, e13580
Journal for ImmunoTherapy of Cancer, 2025, e011611
S5430 Metoprolol Metoprolol is a cardioselective β1-adrenergic blocking agent with log Kd values of −7.26±0.07, −6.89±0.09, −5.16±0.12 for β1, β2, and β3 adrenoceptors, respectively. It is used for acute myocardial infarction, heart failure, angina pectoris and mild to moderate hypertension.
Drug Delivery, November 26 2025, 2585612
Frontiers in Pharmacology, December 06 2022, 1049640
Pharmaceuticals (Basel), 2025, 18(2)181

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