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Adrenergic Receptor Antagonist/Agonists

Other Endocrinology & Hormones Related Inhibitors

Androgen Receptor Estrogen/progestogen Receptor Aromatase 5-alpha Reductase RAAS Glucocorticoid Receptor ACE Mineralocorticoid Receptor PGDS Progesterone Receptor

Isoform-selective Products

Cat.No. Product Name Information Product Use Citations Product Validations
S2521 Epinephrine bitartrate Epinephrine bitartrate (Adrenalinium) is an alpha- and beta-adrenergic receptor stimulator.
Advanced Science, 2025, e13580
iScience, 2024, 27(10):110862
Sci Adv, 2024, 10(33):eado1533
S4076 Propranolol HCl Propranolol HCl (AY-64043, ICI-45520, NCS-91523) is a competitive non-selective beta-adrenergic receptors inhibitor.
Cell Res, 2024, 10.1038/s41422-024-00946-z
J Immunother Cancer, 2024, 12(11)e009805
Sci Rep, 2024, 14(1):4178
S4009 Mirabegron Mirabegron (YM 178) is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.
Biomed Pharmacother, 2025, 183:117816
iScience, 2024, 27(10):110862
J Pers Med, 2022, 12(2)258
S1831 Carvedilol Carvedilol (BM-14190, SKF 105517) is a non-selective beta blocker/alpha-1 blocker, used to treat congestive heart failure (CHF) and high blood pressure.
Communications Medicine, 2025, 420
Gastroenterology, 2024, 167(5):993-1007
J Immunother Cancer, 2024, 12(11)e009805
S8114 ICI 118551 Hydrochloride (Zenidolol) Zenidolol (ICI-118551) Hydrochloride is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
Immunity, 2025, S1074-7613(25)00226-2
Advanced Science, 2025, e13580
Journal for ImmunoTherapy of Cancer, 2025, e011611
S9507 (−)-Norepinephrine (−)-Norepinephrine (Arterenol, Levarterenol, L-Noradrenaline) is a natural neurotransmitter and hormone. It is an agonist of adrenergic receptors with Ki values of 330, 56, and 740 nM for α1, α2, and β1 adrenoceptors, respectively.This compound can be used to induce animal models of Cardiomyopathy.
Drug Design, Development and Therapy, 2025, 4585-4603
Drug Des Devel Ther, 2025, 19:4585-4603
BMC Nephrology, 2025, 498
S2516 Xylazine HCl Xylazine(BAY 1470 hydrochloride) is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant.
J Immunother Cancer, 2024, 12(11)e009805
Cell Death Dis, 2023, 14(5):318
Eur J Pharmacol, 2021, 911:174522
S2569 Phenylephrine HCl Phenylephrine HCl is a selective α1-adrenergic receptor agonist, used primarily as a decongestant.
J Am Heart Assoc, 2025, 14(1):e037400
NPJ Regen Med, 2023, 8(1):9
Front Immunol, 2022, 13:1090773
Verified customer review of Phenylephrine HCl
S5430 Metoprolol Metoprolol is a cardioselective β1-adrenergic blocking agent with log Kd values of −7.26±0.07, −6.89±0.09, −5.16±0.12 for β1, β2, and β3 adrenoceptors, respectively. It is used for acute myocardial infarction, heart failure, angina pectoris and mild to moderate hypertension.
Pharmaceuticals (Basel), 2025, 18(2)181
Drug Metab Dispos, 2025, 53(4):100049
Europace, 2024, euae252
S2507 Salbutamol (Albuterol) Sulfate Salbutamol (Albuterol) Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.
Front Pharmacol, 2025, 16:1621775
Front Physiol, 2022, 13:800055
cell, 2020, 180(1):64-78.e16
Verified customer review of Salbutamol (Albuterol) Sulfate

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