GPCR Compound Library

Catalog No.L2200

Offered in 96 or 384 well plate format

A unique collection of 746 small molecules targeting G protein coupled receptors for high throughput screening (HTS) and high content screening (HCS).

Size Price  
Pre-dissolved In DMSO or Water
USD 8598
USD 12618

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GPCR Compound Library Contents

Cited by 31 Publications

Description & Advantages

•A unique collection of 746 small molecules targeting G protein coupled receptors for high throughput screening (HTS) and high content screening (HCS)
• All of the small molecules in the GPCR library are well characterized with biological and pharmaceutical activity
• A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery
• It is estimated about 200 so-called orphan GPCRs are functionally unknown, as a result, use of our GPCR Small Molecule Compound Library for screening the functionally unknown GPCRs may yield potentially new GPCR-based drug candidates
• The GPCR compound library contains small molecules associated with receptors including 5-HT Receptor, Dopamine Receptor, Opioid Receptor, Adrenergic Receptors, Cannabinoid Receptor, mGluR, and ETA-receptor etc.
• Structurally diverse, medicinally active, and cell permeable
• Rich documentation with structure and customer reviews
• NMR and HPLC validated to ensure the highest purity

Product Details

Formulation: 676 compounds pre-dissolved in 10mM DMSO, 46 compounds pre-dissolved in 10mM water, 20 compounds pre-dissolved in 2mM DMSO and 4 compounds pre-dissolved in 2mM water
Container: 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Stability: in DMSO
in DMSO
Shipping: Blue ice or dry ice
Packaging: Inert gas

GPCR Compound Library Composition

HTS Facility Partners

See Other Libraries