Inhibitor Library

Catalog No.L1100

Offered in 96 or 384 well plate format

A unique collection of 2771 inhibitors for high throughput screening (HTS) and high content screening (HCS).

Size

Price

Pre-dissolved In DMSO or Water
100uL/well (2mM or 10mM solution)	USD 24274
2x100uL/well (2mM or 10mM solution)	USD 44451

Selleck USA Tel: (832) 582-8158 [email protected]

You Could Select:

Specific Compounds Quantities Plate Map Dry/solid or DMSO solution

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Inhibitor Library Contents

Download the Inhibitor Library - SDF

Download the Inhibitor Library - XLSX

Cited by 39 Publications

Nat Med,2017,23(4):405-408

PubMed: 28388612 ( click the link to review the publication )

Nat Med,2014,20(8):954-60

PubMed: 24997607 ( click the link to review the publication )

Sci Adv,2019,5(6):eaav9784

PubMed: 31249867 ( click the link to review the publication )

Neuropsychopharmacology,2019,10.1038/s41386-018-0266-7

PubMed: 30518933 ( click the link to review the publication )

Breast Cancer Res,2019,21(1):37

PubMed: 30845991 ( click the link to review the publication )

Endocr Relat Cancer,2019,10.1530/ERC-18-0509

PubMed: 30730850 ( click the link to review the publication )

Neurobiol Aging,2019,76:24-34

PubMed: 30640040 ( click the link to review the publication )

Cancer Manag Res,2019,11:8391-8405

PubMed: 31571995 ( click the link to review the publication )

Acta Pharmacol Sin,2019,10.1038/s41401-019-0246-4

PubMed: 31197246 ( click the link to review the publication )

BMC Cancer,2019,19(1):102

PubMed: 30678647 ( click the link to review the publication )

Bioengineered,2019,10(1):98-107

PubMed: 31023186 ( click the link to review the publication )

Kaohsiung J Med Sci,2019,10.1002/kjm2.12051

PubMed: 30896891 ( click the link to review the publication )

Cell Rep,2018,22(5):1185-1199

PubMed: 29386107 ( click the link to review the publication )

Endocr Relat Cancer,2018,25(3):367-380

PubMed: 29444910 ( click the link to review the publication )

Mol Oncol,2018,12(9):1526-1539

PubMed: 30055072 ( click the link to review the publication )

Cancer Sci,2018,109(4):1220-1229

PubMed: 29453896 ( click the link to review the publication )

Sci Rep,2018,8(1):13106

PubMed: 30166612 ( click the link to review the publication )

J Cell Physiol,2018,233(1):422-433

PubMed: 28294327 ( click the link to review the publication )

Cancer Immunol Res,2017,5(9):790-803

PubMed: 28775208 ( click the link to review the publication )

Anal Chem,2017,89(12):6678-6685

PubMed: 28520400 ( click the link to review the publication )

Mol Cancer Ther,2017,16(9):1739-1750

PubMed: 28572168 ( click the link to review the publication )

Antimicrob Agents Chemother,2017,62(1)

PubMed: 29061736 ( click the link to review the publication )

Sci Rep,2017,7(1):14341

PubMed: 29085027 ( click the link to review the publication )

Pharmacol Res,2016,113(Pt A):216-227

PubMed: 27543462 ( click the link to review the publication )
PLoS One,2016,11(2):e0149848

PubMed: 26919709 ( click the link to review the publication )

Sensors (Basel),2016,16(3)

PubMed: 26999137 ( click the link to review the publication )

Sci Rep,2016,6:25694

PubMed: 27157787 ( click the link to review the publication )

Oncotarget,2016,7(3):2545-54

PubMed: 26575423 ( click the link to review the publication )

Clin Cancer Res,2015,21(5):1172-82

PubMed: 25549722 ( click the link to review the publication )

Biosens Bioelectron,2015,68:699-704

PubMed: 25668591 ( click the link to review the publication )

Mol Cancer Ther,2015,14(5):1213-23

PubMed: 25777964 ( click the link to review the publication )

Cell Cycle,2015,14(1):109-22

PubMed: 25602521 ( click the link to review the publication )

PLoS One,2015,10(11):e0142655

PubMed: 26569102 ( click the link to review the publication )

Oncotarget,2015,6(3):1531-43

PubMed: 25605238 ( click the link to review the publication )

Head Neck,2015,37(12):1722-32

PubMed: 24986420 ( click the link to review the publication )

Mol Cancer Res,2014,12(5):703-13

PubMed: 24554781 ( click the link to review the publication )

Oncotarget,2014,5(15):6512-25

PubMed: 25156567 ( click the link to review the publication )

Curr Protoc Chem Biol,2014,4:177-191

PubMed: 26705509 ( click the link to review the publication )

Description & Advantages

• A unique collection of 2771 small molecule inhibitors for high throughput screening (HTS) and high content screening (HCS)

• Includes most Selleck inhibitors, APIs, natural products, and chemotherapeutic agents

• Some inhibitors have been approved by the FDA

• Targets PI3K, VEGFR, and RTK pathway, HDAC, Aurora Kinase, CDK and Cell Cycle regulators, Integrase/Proteasome, Phosphatase etc

• Structurally diverse, medicinally active, and cell permeable

• Rich documentation with structure, IC50, and customer reviews

• NMR and HPLC validated to ensure high purity

Product Details

Formulation:	2582 compounds pre-dissolved in 10mM DMSO, 96 compounds pre-dissolved in 10mM water, 87 compounds pre-dissolved in 2mM DMSO and 6 compounds pre-dissolved in 2mM water
Container:	96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Stability:	12 months -20°C in DMSO
Stability:	24 months -80°C in DMSO
Shipping:	Blue ice or dry ice
Packaging:	Inert gas

Inhibitor Library Composition

HTS Facility Partners

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