β-adrenergic receptor Selective Inhibitors | Agonists | Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S4085 Levobetaxolol HCl

Levobetaxolol exhibits a higher affinity at cloned human β1 and β2 receptors with Ki value of 0.76 nM and 32.6 nM, respectively.

Selective β2-adrenergic receptor, Ki: 32.6 nM; β1-adrenergic receptor, Ki: 0.76 nM; β2-adrenergic receptor, Ki: 32.6 nM; β1-adrenergic receptor, Ki: 0.76 nM
S1549 Nebivolol

Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.

Selective β1-adrenoceptor, IC50: 0.8 nM
S4123 Timolol Maleate

Timolol Maleate is a non-selective, beta-adrenergic receptor antagonist for β1/β2 with Ki of 1.97 nM/2.0 nM.

Selective β2-adrenergic receptor, Ki: 2.0 nM; β1-adrenergic receptor, Ki: 1.97 nM
S2507 Salbutamol Sulfate

Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.

Selective β2-adrenergic receptor, IC50: 8930 nM; β2-adrenergic receptor, IC50: 8.93 nM
S4076 Propranolol HCl

Propranolol HCl is a competitive non-selective beta-adrenergic receptors inhibitor with IC50 of 12 nM.

Selective β-adrenergic receptor, IC50: 12 nM
S4009 Mirabegron

Mirabegron is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.

Selective β3-adrenoceptor, EC50: 22.4 nM
S3083 Indacaterol Maleate

Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.

Selective β-adrenoceptor, pKi: 7.36
S4127 Terbutaline Sulfate

Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM.

Selective β2-adrenergic receptor, IC50: 53 nM
S1827 Betaxolol HCl

Betaxolol is a β1 adrenergic receptor blocker with IC50 of 6 μM.

Selective β1-adrenergic receptor, IC50: 6 μM
S4277 Bambuterol HCl

Bambuterol HCl is a potent β-adrenoceptor agonist, used in the treatment of asthma.

Selective
S4010 Acebutolol HCl

Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.

Selective
S4135 Clorprenaline HCl

Clorprenaline HCl is a β2-receptor agonist, it has a significant expansion of the bronchial effect.

Selective
S1206 Bisoprolol fumarate

Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker.

Selective
S2566 Isoprenaline HCl

Isoprenaline is a non-selective beta-adrenergic receptor agonist, used for the treatment of bradycardia and heart block.

Selective
S2509 Sotalol

Sotalol is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM.

Selective
S4100 Esmolol HCl

Esmolol is a cardioselective b-blocker, used to control rapid heartbeats or abnormal heart rhythms.

Selective
S4278 Carteolol HCl

Carteolol HCl is a β-adrenoceptor antagonist, used for the treatment of glaucoma.

Selective
S2091 Betaxolol

Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.

Selective
S4296 Salmeterol Xinafoate

Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms.

Selective
S2020 Formoterol Hemifumarate

Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist to β2 and β1 receptors with pKd of 8.12 and 5.58, respectively.

Selective
S2533 Ritodrine HCl

Ritodrine HCl is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist.

Selective
S1856 Metoprolol Tartrate

Metoprolol Tartrate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL.

Selective
S2691 BMY 7378 Dihydrochloride

BMY 7378 is a multi-targeted inhibitor of α2C-adrenoceptor and α1D-adrenoceptor with pKi of 6.54 and 8.2, respectively, and acts as a mixed agonist and antagonist for 5-HT1A receptor with pKi of 8.3.

Pan β2-adrenoceptor, pIC50: <5.0; β1-adrenoceptor, pIC50: 5.1
S2521 Epinephrine Bitartrate

Epinephrine Bitartrate is an alpha- and beta-adrenergic receptor stimulator.

Pan
S4291 Labetalol HCl

Labetalol HCl is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors, used in the treatment of high blood pressure.

Pan
S1831 Carvedilol

Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.

Pan