PPARα Selective Inhibitors | Activators | Agonists | Antagonists
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
|S8029||WY-14643 (Pirinixic Acid)||
WY 14643 (Pirinixic Acid) is a potent peroxisome proliferator and activator of PPARα with EC50 of 1.5 μM.
|Selective||PPARα, EC50: 1.5 μM|
Clofibric acid is a PPARα agonist and hypolipidemic agent.
Gemfibrozil (Lopid) is a compound used to lower lipid levels.
Fenofibrate (Tricor, Trilipix) is a compound of the fibrate class and fibric acid derivative.
GW9662 is a selective PPAR antagonist for PPARγ with IC50 of 3.3 nM, with at least 100 to 1000-fold functional selectivity in cells with PPARγ versus PPARα and PPARδ.
|Pan||PPARα, IC50: 32 nM|
T0070907 is a potent and selective PPARγ inhibitor with IC50 of 1 nM, with a >800-fold selectivity over PPARα and PPARδ.
|Pan||PPARα, IC50: 0.85 μM|
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