NMDA receptor Selective Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S2857 MK-801 (Dizocilpine)

MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.

Selective NMDA Receptor, Ki: 30.5 nM
S2876 (-)-MK 801 Maleate

MK-801 is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.

Selective NMDA Receptor, Kd: 37.2 nM
S4091 Ifenprodil Tartrate

Ifenprodil is an atypical noncompetitive antagonist at the NMDA receptor, it interacts with high affinity at a homogeneous population of NMDA receptors in neonatal rat forebrain with IC50 of 0.3 μM.

Selective NMDA Receptor, IC50: 0.3 μM
S7072 NMDA (N-Methyl-D-aspartic acid)

NMDA(N-Methyl-D-aspartic acid)is a specific agonist for NMDA receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor. Phase 4.

S1614 Riluzole

Riluzole is a drug used to treat amyotrophic lateral sclerosis.