nAChR Selective Inhibitors | Agonists | Modulators

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S4162 Benzethonium Chloride

Benzethonium chloride is a potent inhibitor of nAChRs, it inhibits α4β2 nAChRs and α7 nAChRs with IC50 of 49 nM and 122 nM, respectively.

Selective α7 nAChRs, IC50: 122 nM; α4β2 nAChRs, IC50: 49 nM
S2629 PNU-120596

PNU-120596 is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.

Selective α7 nAChR, EC50: 216 nM
S4072 Decamethonium Bromide

Decamethonium Bromide is a nicotinic AChR partial agonist and neuromuscular blocking agent.

Selective
S4121 Succinylcholine Chloride Dihydrate

Succinylcholine Chloride Dihydrate is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.

Selective
S2287 Cytisine

Cytisine is a nicotinic acetylcholine receptor agonist.

Selective