GABAA receptor Selective Agonists | Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S7071 (+)-Bicuculline

(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.

Selective GABAA receptor, IC50: 2 μM
S1332 Flumazenil

Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses.

S2399 Dihydromyricetin

Dihydromyricetin (Ampelopsin, Ampeloptin) is a natural antioxidant flavonoid from Ampelopsis grossedentata.

S2269 Baicalin

Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors.

S1329 Etomidate

Etomidate is a GABAA receptor agonist, used as a short-acting anaesthetic agent or sedative.

S4197 Bemegride

Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning.