HomeNew GABA Receptor Inhibitors

New GABA Receptor Inhibitors

Catalog No. Product Name Information
E6042 Riluzole hydrochloride Riluzole hydrochloride (PK 26124 hydrochloride) is an antiepileptic drug, a state-dependent inhibitor of Na+ channels and a selective inhibitor of glutamate release. It also inhibits GABA uptake with an IC50 of 43 µM.
F2491 GABA B Receptor 2/GABBR2 Rabbit mAb GABA B Receptor 2/GABBR2,GABA(B)R2
E4920 Baclofen hydrochloride Baclofen hydrochloride is an agonist of the GABAB receptor that mimics the action of GABA, leading to slow presynaptic inhibition via the GABAB receptor. It improves the function of the ubiquitin-proteasome system (UPS) and enhances cell survival in both in vitro and in vivo models of Huntington's disease (HD).
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