P2Y receptor Selective Inhibitors | Antagonists | Modulators

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S4079 Ticagrelor

Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist with Ki of 2 nM.

Selective P2Y12, Ki: 2 nM
S2855 MRS 2578

MRS2578 is a potent P2Y6 receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors.

Selective P2Y6, IC50: 37 nM
S1415 Clopidogrel

Clopidogrel is an oral, thienopyridine class antiplatelet agent.

S1258 Prasugrel

Prasugrel is a thienopyridine ADP receptor (P2Y12) antagonist, used for the reduction of thrombotic cardiovascular events.