H3 receptor Selective Inhibitors | Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S2813 Ciproxifan

Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.

 Selective Histamine H3 receptor, IC50: 9.2 nM
S3176 Betahistine 2HCl

Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM.

 Selective Histamine H3 receptor, IC50: 1.9 μM