PKM

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S8616 PKM2 inhibitor(compound 3k) <1 mg/mL 6 mg/mL <1 mg/mL
S7928 DASA-58 <1 mg/mL 91 mg/mL <1 mg/mL
S5545 DL-Serine 8 mg/mL <1 mg/mL -1 mg/mL
Catalog No. Information Product Use Citations Product Validations
S8616New

PKM2 inhibitor(compound 3k)

PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.

S7928

DASA-58

DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator.

S5545New

DL-Serine

Serine is a non-essential amino acid and a natural ligand and allosteric activator of pyruvate kinase M2.

Tags: PKM activator | PKM inhibitor | PKM modulator |PKM activity