FAAH
Signaling Pathway Map
Research Area
Inhibitory Selectivity
FAAH Products
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S2631 |
URB597URB597 is a potent, orally bioavailable FAAH inhibitor with IC50 of 4.6 nM, with no activity on other cannabinoid-related targets. Phase 1. |
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| S2666 |
PF-3845PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2. |
||
| S5329New |
FAAH-IN-2FAAH-IN-2 is an inhibitor of fatty acid amide hydrolase (FAAH). |
||
| S2377 |
Biochanin ABiochanin A, an O-methylated isoflavone from Trifolium pratense, inhibits protein tyrosine kinase (PTK) of epidermal growth factor receptor with IC50 values of 91.5 μM. |
||
| S2828 |
JNJ-1661010JNJ-1661010 is a potent and selective FAAH inhibitor with IC50 of 10 nM (rat) and 12 nM (human), exhibits >100-fold selectivity for FAAH-1 when compared to FAAH-2. |
||
| S5932New |
BIA 10-2474BIA 10-2474 is a novel fatty acid amide hydrolase (FAAH) inhibitor, with a potent inhibitory effect upon FAAH and prolonged action in vivo. |
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S2631 |
URB597URB597 is a potent, orally bioavailable FAAH inhibitor with IC50 of 4.6 nM, with no activity on other cannabinoid-related targets. Phase 1. |
||
| S2666 |
PF-3845PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2. |
||
| S5329New |
FAAH-IN-2FAAH-IN-2 is an inhibitor of fatty acid amide hydrolase (FAAH). |
||
| S2377 |
Biochanin ABiochanin A, an O-methylated isoflavone from Trifolium pratense, inhibits protein tyrosine kinase (PTK) of epidermal growth factor receptor with IC50 values of 91.5 μM. |
||
| S2828 |
JNJ-1661010JNJ-1661010 is a potent and selective FAAH inhibitor with IC50 of 10 nM (rat) and 12 nM (human), exhibits >100-fold selectivity for FAAH-1 when compared to FAAH-2. |
||
| S5932New |
BIA 10-2474BIA 10-2474 is a novel fatty acid amide hydrolase (FAAH) inhibitor, with a potent inhibitory effect upon FAAH and prolonged action in vivo. |
