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AdipoR

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Cat.No. Product Name Information Product Use Citations Product Validations
S7365 AdipoRon AdipoRon (SC-396658) is a novel, and orally bioavailable adiponectin receptor agonist with KD of 1.8 and 3.1 μM for AdipoR1 and AdipoR2, respectively.
Aging Cell, 2025, 24(2):e14390
Sci Adv, 2025, 11(29):eadv6642
Environ Health Perspect, 2024, 132(11):117003
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S4738 Arctiin Arctiin (Arctigenin-4-Glucoside, NSC 315527) acts on an agonists of the adiponectin receptor 1 with anti-cancer effects.
The American Journal of Chinese Medicine, March 14, 2024, 471-492
Biochemical Pharmacology, March 1, 2026, 117691
S3822 Schisandrin A Schisandrin A (Sch A, Deoxyschizandrin, Wuweizisu A) is an active component of Schisandrae Fructus with liver-protective, antitumor, and antioxidant activities. It is an agonist of the adiponectin receptor 2 (AdipoR2) with the IC50 value of 3.5 μM.
S2304 Gramine Gramine (Donaxine) is a natural indole alkaloid isolated from giant reed, acts as an active adiponectin receptor (AdipoR) agonist, with IC50 of 3.2 µM and 4.2 µM for AdipoR2 and AdipoR1, respectively. This compound is also a human and mouse β2-Adrenergic receptor (β2-AR) agonist.
Journal of Cellular and Molecular Medicine, 2021 Jul 19, 7980-7992
Journal of Cellular and Molecular Medicine, 2021, 7980-7992