- δ-opioid receptor
- κ-opioid receptor
- μ-opioid receptor
mumumu-opioid-receptor Selective Inhibitors | Agonists | Antagonists
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
Naltrexone HCl is an opioid receptor antagonist with IC50 of 8 nM used primarily in the management of alcohol dependence and opioid dependence.
|Selective||opioid receptor, IC50: 8 nM|
Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM.
Racecadotril is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM
Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose.
Loperamide HCl is an opioid-receptor agonist with an ED50 of 0.15 mg/kg.
ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel. Phase 2.
|Pan||μ-opioid receptor, Ki: 32 nM|
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