Home GPCR & G Protein PAR PAR2 Selective Inhibitors | Antagonists

PAR2 Selective Inhibitors | Antagonists

  • PAR1
  • PAR2
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S9744 AZ3451 AZ3451 is a potent antagonist of protease-activated receptor 2 (PAR2) that binds to a remote allosteric site outside the helical bundle with IC50 of 23 nM. Selective PAR2, IC50: 23 nM
S9915 FSLLRY-NH2 TFA FSLLRY-NH2 TFA (FSY-NH2) is a selective protease-activated receptor 2 (PAR2) inhibitor with an ic50 of 50 µM in PAR2-KNRK cells. Selective