- OX1 receptor
- OX2 receptor
OX1 receptor Selective Antagonists
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.
|Selective||OX1 (membrane), Ki: 27 nM; OX1 (whole cell), Ki: 57 nM|
SB-334867 is a selective orexin-1 (OX1) receptor antagonist.
Almorexant HCl (ACT-078573) is an orally active, dual orexin receptor antagonist with IC50 of 6.6 nM and 3.4 nM for OX1 and OX2 receptor, respectively. Phase 3.
|Pan||OX1 receptor, IC50: 6.6 nM|
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