Home GPCR & G Protein Adenosine Receptor Adenosine-A1-receptor Selective Antagonists

Adenosine-A1-receptor Selective Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S0272 Derenofylline (SLV320) Derenofylline (SLV320) is a selective and potent adenosine A1 antagonist with Ki of 1 nM. Derenofylline shows selective for adenosine A1 over A2A, A2B, and A3 receptors with Ki of 398 nM, 3981 nM, and 200 nM, respectively. Selective Adenosine A1 receptor, Ki: 1 nM