New Histamine Receptor Antagonists

Catalog No. Product Name Information
E7924 GSK189254A GSK189254A (GSK189254 free base) is a histamine H3 receptor antagonist with pKi values of 9.59-9.90 for human H3 and 8.51-9.17 for rat H3.
E6055 Epinastine Epinastine (WAL801) is potent nonsedative antiallergic agent and an antagonist of histamine H1 receptor. It inhibits the actions of leukotrienes, platelet-activating factor (PAF), and bradykinin. It also stabilizes mast cells and reduces IL-8 release from eosinophils, helping to control allergic inflammation.
All Histamine Receptor Antagonists