NAMPT

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S7316 STF-118804 <1 mg/mL 61 mg/mL <1 mg/mL
S8444 KPT-9274 <1 mg/mL 100 mg/mL 100 mg/mL
S8117 GMX1778 (CHS828) <1 mg/mL 74 mg/mL <1 mg/mL
S7968 P7C3 <1 mg/mL 95 mg/mL 20 mg/mL
Catalog No. Information Product Use Citations Product Validations
S7316

STF-118804

STF-118804 is a highly specific NAMPT inhibitor.

S8444New

KPT-9274

KPT-9274 is an orally bioavailable small molecule that is a non-competitive dual inhibitor of PAK4 and NAMPT. It shows an IC50 of ~120 nM for NAMPT in a cell-free enzymatic assay.

S8117

GMX1778 (CHS828)

GMX1778 (CHS828) is a potent and specific inhibitor of nicotinamide phosphoribosyltransferase (NAMPT) with IC50 and Kd of < 25 nM and 120 nM, respectively. Phase 1.

S7968

P7C3

P7C3 is a potent proneurogenic and neuroprotective chemical that targets NAMPT enzyme.