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CRT0066101

Name: CRT0066101
Brand: Selleck Chemicals
SKU: S3414
Rating: 5 (3 reviews)

Catalog No.S3414

For research use only.

CRT0066101 is a specific inhibitor of all Protein kinase D (PKD) isoforms.

CAS No. 956121-30-5

Selleck's CRT0066101 has been cited by 3 Publications

Purity & Quality Control

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Download Inhibitor Catalog

Biological Activity

Description	CRT0066101 is a specific inhibitor of all Protein kinase D (PKD) isoforms.

Protocol (from reference)

Chemical Information

Molecular Weight
Formula
CAS No.	956121-30-5
Storage	3 years	-20°C	powder
Storage	2 years	-80°C	in solvent

In vivo Formulation Calculator (Clear solution)

Step 1: Enter information below (Recommended: An additional animal making an allowance for loss during the experiment)

Dosage: mg/kg Average weight of animals: g Dosing volume per animal:μL Number of animals:

Step 2: Enter the in vivo formulation (This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO + % + % Tween 80 + % ddH₂O

%DMSO+ %

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH₂O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such
as vortex, ultrasound or hot water bath can be used to aid dissolving.

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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