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PPMTase

Inhibitory Selectivity

PPMTase Products

All (1) PPMTase Inhibitors (1)

Catalog No.	Information	Product Use Citations	Product Validations
S7684	Salirasib Salirasib (Farnesylthiosalicylic acid, FTS) is a potent competitive prenylated protein methyltransferase (PPMTase) inhibitor with K_i of 2.6 μM, which inhibits _Ras methylation. Salirasib exerts antitumor effects and induces autophagy. Salirasib exerts antitumor effects and induces autophagy. Phase 2.	Mol Oncol, 2018, 12(2):224-238 Food Chem Toxicol, 2018, 119:464-478 Oncotarget, 2017, 8(30):49824-49838

Catalog No.

Information

Product Use Citations

Product Validations

S7684

Salirasib

Salirasib (Farnesylthiosalicylic acid, FTS) is a potent competitive prenylated protein methyltransferase (PPMTase) inhibitor with K_i of 2.6 μM, which inhibits _Ras methylation. Salirasib exerts antitumor effects and induces autophagy. Salirasib exerts antitumor effects and induces autophagy. Phase 2.

Mol Oncol, 2018, 12(2):224-238

Food Chem Toxicol, 2018, 119:464-478

Oncotarget, 2017, 8(30):49824-49838

Catalog No.	Information	Product Use Citations	Product Validations
S7684	Salirasib Salirasib (Farnesylthiosalicylic acid, FTS) is a potent competitive prenylated protein methyltransferase (PPMTase) inhibitor with K_i of 2.6 μM, which inhibits _Ras methylation. Salirasib exerts antitumor effects and induces autophagy. Salirasib exerts antitumor effects and induces autophagy. Phase 2.	Mol Oncol, 2018, 12(2):224-238 Food Chem Toxicol, 2018, 119:464-478 Oncotarget, 2017, 8(30):49824-49838