PPMTase
Inhibitory Selectivity
PPMTase Products
Catalog No. | Information | Product Use Citations | Product Validations |
---|---|---|---|
S7684 |
SalirasibSalirasib (Farnesylthiosalicylic acid, FTS) is a potent competitive prenylated protein methyltransferase (PPMTase) inhibitor with Ki of 2.6 μM, which inhibits Ras methylation. Salirasib exerts antitumor effects and induces autophagy. Salirasib exerts antitumor effects and induces autophagy. Phase 2. |
Catalog No. | Information | Product Use Citations | Product Validations |
---|---|---|---|
S7684 |
SalirasibSalirasib (Farnesylthiosalicylic acid, FTS) is a potent competitive prenylated protein methyltransferase (PPMTase) inhibitor with Ki of 2.6 μM, which inhibits Ras methylation. Salirasib exerts antitumor effects and induces autophagy. Salirasib exerts antitumor effects and induces autophagy. Phase 2. |