GlyR

Other Transmembrane Transporters Related Inhibitors

CFTR CRM1 Calcium Channel Proton Pump P-gp Sodium Channel ATPase Potassium Channel CD markers GLUT

Cat.No.	Product Name	Information	Product Use Citations
S0920	Ginkgolide J	Ginkgolide J is a minor constituent of terpene trilactone mixture of Ginkgo biloba leaves extract that inhibits GlyR-operated channels with IC50 of 2.0 μM. This compound also inhibits cell death of rodent hippocampal neurons caused by Aβ1–42. It exhibits anti‑inflammatory activity.
S9294	Gelsemine	Gelsemine, a principal alkaloid from Gelsemium sempervirens Ait., is a highly toxic compound and may be a glycine receptor agonist with significantly higher binding affinity for some of these receptors than its native agonist, glycine.
S6172	Brucine sulfate heptahydrate	Brucine is an alkaloid that acts as an antagonist at glycine receptors and paralyzes inhibitory neurons.	Sci Rep, 2023, 13(1):18492.
S6100	Picrotoxin	Picrotoxin (Picrotin, Cocculin, Cocculus, NSC 403139), a plant alkaloid, is a non-competitive antagonist of neuronal GABA and glycine receptors.This product is a hazardous chemical (acute toxicity/flammable/skin corrosive). Please use it while wearing a protective face mask, gloves, and clothing.