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S1191
|
Fulvestrant (Faslodex) |
Fulvestrant is an estrogen receptor (ER) antagonist with IC50 of 0.094 nM. |
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S1972
|
Tamoxifen Citrate (Nolvadex) |
Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding. |
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S1227
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Evista(Raloxifene HCl) |
Raloxifene is estrogen antagonists, inhibits human cytosolic aldehyde oxidase-catalyzed phthalazine oxidation activity with IC50 of 5.7 nM. |
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S1776
|
Toremifene Citrate (Fareston, Acapodene) |
Toremifene Citrate(Fareston, Acapodene) is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. |
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S2606
|
Mifepristone (Mifeprex) |
Mifepristone (Mifeprex, RU-486, RU-38486, Mifegyne) is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. |
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S2128
|
Bazedoxifene HCl |
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM. |
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S1251
|
Dienogest |
Dienogest is an orally active synthetic progesterone (or progestin). |
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S1598
|
LY500307 (Erteberel) |
LY500307 (SERBA-1) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM. |
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S2832
|
Epiandrosterone (3β-androsterone) |
Epiandrosterone (3β-androsterone) is a steroid hormone with weak androgenic activity which acts as a L-type Ca2+ channel antagonist. |
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S1914
|
Pregnenolone |
Pregnenolone is an endogenous steroid hormone for inhibition of M1 receptor- and M3 receptor-mediated currents with IC50 of 11.4 µM and 6.0 µM, respectively.
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S2611
|
Ethisterone |
Ethisterone is a progestogen hormone being considered to treat prostate cancer.
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S2450
|
Equol |
Equol is an isoflavandiol metabolized from daidzein by bacterial flora in the intestines. |
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S3160
|
Ethynodiol diacetate |
Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills. |
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S3149
|
Estradiol valerate |
Estradiol is a synthetic ester used to treat menopausal symptoms and hormone deficiencies. |
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S3167
|
Altrenogest |
Altrenogest is a progestogen structurally related to veterinary steroid trenbolone. |
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S2567
|
Medroxyprogesterone acetate |
Medroxyprogesterone acetate is a progestin, a synthetic variant of the human hormone progesterone and a potent progesterone receptor agonist. |
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S2561
|
Clomifene citrate (Serophene) |
Clomifene citrate (Serophene) is a selective estrogen receptor modulator. |
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S2473
|
Hexestrol(Bibenzyl) |
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively. |
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S2466
|
Estriol |
Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells. |
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S2167
|
Bazedoxifene acetate |
Bazedoxifene is a third generation selective estrogen receptor modulator (SERM). |
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S1665
|
Estrone |
Estrone is an estrogenic hormone. |
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S1377
|
Drospirenone |
Drospirenone is a synthetic progestin that is an analog to spironolactone. |
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S1376
|
Gestodene |
Gestodene is a progestogen hormonal contraceptive. |
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S1238
|
Nolvadex |
Tamoxifen is an antagonist of the estrogen receptor in breast tissue. |
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