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Estrogen/progestogen Receptor

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Cat.No.	Product Name	Solubility (25°C)
S1191	Fulvestrant (Faslodex)	<1 mg/mL	121 mg/mL	121 mg/mL
S1972	Tamoxifen Citrate (Nolvadex)	<1 mg/mL	113 mg/mL	<1 mg/mL
S1227	Evista(Raloxifene HCl)	<1 mg/mL	102 mg/mL	<1 mg/mL
S1776	Toremifene Citrate (Fareston, Acapodene)	<1 mg/mL	120 mg/mL	<1 mg/mL
S2606	Mifepristone (Mifeprex)	<1 mg/mL	86 mg/mL	19 mg/mL
S2128	Bazedoxifene HCl	<1 mg/mL	101 mg/mL	<1 mg/mL
S1251	Dienogest	<1 mg/mL	62 mg/mL	5 mg/mL
S1598	LY500307 (Erteberel)	<1 mg/mL	57 mg/mL	57 mg/mL
S1377	Drospirenone	<1 mg/mL	73 mg/mL	11 mg/mL
S1376	Gestodene	<1 mg/mL	62 mg/mL	8 mg/mL
S1665	Estrone	<1 mg/mL	54 mg/mL	<1 mg/mL
S2466	Estriol	<1 mg/mL	57 mg/mL	10 mg/mL
S2473	Hexestrol(Bibenzyl)	<1 mg/mL	42 mg/mL	42 mg/mL
S2450	Equol	<1 mg/mL	48 mg/mL	48 mg/mL
S2561	Clomifene citrate (Serophene)	<1 mg/mL	120 mg/mL	11 mg/mL
S2567	Medroxyprogesterone acetate	<1 mg/mL	12 mg/mL	12 mg/mL
S2611	Ethisterone	<1 mg/mL	0.05 mg/mL	<1 mg/mL
S1914	Pregnenolone	<1 mg/mL	22 mg/mL	22 mg/mL
S2832	Epiandrosterone (3β-androsterone)	<1 mg/mL	58 mg/mL	58 mg/mL
S3167	Altrenogest	<1 mg/mL	62 mg/mL	2 mg/mL
S3149	Estradiol valerate	<1 mg/mL	71 mg/mL	<1 mg/mL
S3160	Ethynodiol diacetate	77 mg/mL	77 mg/mL	<1 mg/mL

Estrogen/progestogen Receptor Chemicals (24)
water-soluble

Cat.No.	Product Name	Information	Product Citations
S1191	Fulvestrant (Faslodex)	Fulvestrant is an estrogen receptor (ER) antagonist with IC50 of 0.094 nM.	PLoS One, 2011, 6(7):e21112
S1972	Tamoxifen Citrate (Nolvadex)	Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding.
S1227	Evista(Raloxifene HCl)	Raloxifene is estrogen antagonists, inhibits human cytosolic aldehyde oxidase-catalyzed phthalazine oxidation activity with IC50 of 5.7 nM.
S1776	Toremifene Citrate (Fareston, Acapodene)	Toremifene Citrate(Fareston, Acapodene) is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body.
S2606	Mifepristone (Mifeprex)	Mifepristone (Mifeprex, RU-486, RU-38486, Mifegyne) is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively.
S2128	Bazedoxifene HCl	Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM.
S1251	Dienogest	Dienogest is an orally active synthetic progesterone (or progestin).
S1598	LY500307 (Erteberel)	LY500307 (SERBA-1) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM.
S1377	Drospirenone	Drospirenone is a synthetic progestin that is an analog to spironolactone.
S1376	Gestodene	Gestodene is a progestogen hormonal contraceptive.

Cat.No.	Product Name	Information
S1665	Estrone	Estrone is an estrogenic hormone.
S2466	Estriol	Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.
S2473	Hexestrol(Bibenzyl)	Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
S2450	Equol	Equol is an isoflavandiol metabolized from daidzein by bacterial flora in the intestines.
S1238	Nolvadex	Tamoxifen is an antagonist of the estrogen receptor in breast tissue.
S2167	Bazedoxifene acetate	Bazedoxifene is a third generation selective estrogen receptor modulator (SERM).
S2561	Clomifene citrate (Serophene)	Clomifene citrate (Serophene) is a selective estrogen receptor modulator.
S2567	Medroxyprogesterone acetate	Medroxyprogesterone acetate is a progestin, a synthetic variant of the human hormone progesterone and a potent progesterone receptor agonist.
S2611	Ethisterone	Ethisterone is a progestogen hormone being considered to treat prostate cancer.
S1914	Pregnenolone	Pregnenolone is an endogenous steroid hormone for inhibition of M1 receptor- and M3 receptor-mediated currents with IC50 of 11.4 µM and 6.0 µM, respectively.

Cat.No.	Product Name	Information
S2832	Epiandrosterone (3β-androsterone)	Epiandrosterone (3β-androsterone) is a steroid hormone with weak androgenic activity which acts as a L-type Ca²⁺ channel antagonist.
S3167	Altrenogest	Altrenogest is a progestogen structurally related to veterinary steroid trenbolone.
S3149	Estradiol valerate	Estradiol is a synthetic ester used to treat menopausal symptoms and hormone deficiencies.
S3160	Ethynodiol diacetate	Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills.

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Estrogen/progestogen Receptor

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Estrogen/progestogen Receptor Chemicals (24)
water-soluble

Cat.No.	Product Name	Solubility (25°C)
Cat.No.	Product Name	Water	DMSO	Ethanol
S1191	Fulvestrant (Faslodex)	<1 mg/mL	121 mg/mL	121 mg/mL
S1972	Tamoxifen Citrate (Nolvadex)	<1 mg/mL	113 mg/mL	<1 mg/mL
S1227	Evista(Raloxifene HCl)	<1 mg/mL	102 mg/mL	<1 mg/mL
S1776	Toremifene Citrate (Fareston, Acapodene)	<1 mg/mL	120 mg/mL	<1 mg/mL
S2606	Mifepristone (Mifeprex)	<1 mg/mL	86 mg/mL	19 mg/mL
S2128	Bazedoxifene HCl	<1 mg/mL	101 mg/mL	<1 mg/mL
S1251	Dienogest	<1 mg/mL	62 mg/mL	5 mg/mL
S1598	LY500307 (Erteberel)	<1 mg/mL	57 mg/mL	57 mg/mL
S1377	Drospirenone	<1 mg/mL	73 mg/mL	11 mg/mL
S1376	Gestodene	<1 mg/mL	62 mg/mL	8 mg/mL
S1665	Estrone	<1 mg/mL	54 mg/mL	<1 mg/mL
S2466	Estriol	<1 mg/mL	57 mg/mL	10 mg/mL
S2473	Hexestrol(Bibenzyl)	<1 mg/mL	42 mg/mL	42 mg/mL
S2450	Equol	<1 mg/mL	48 mg/mL	48 mg/mL
S2561	Clomifene citrate (Serophene)	<1 mg/mL	120 mg/mL	11 mg/mL
S2567	Medroxyprogesterone acetate	<1 mg/mL	12 mg/mL	12 mg/mL
S2611	Ethisterone	<1 mg/mL	0.05 mg/mL	<1 mg/mL
S1914	Pregnenolone	<1 mg/mL	22 mg/mL	22 mg/mL
S2832	Epiandrosterone (3β-androsterone)	<1 mg/mL	58 mg/mL	58 mg/mL
S3167	Altrenogest	<1 mg/mL	62 mg/mL	2 mg/mL
S3149	Estradiol valerate	<1 mg/mL	71 mg/mL	<1 mg/mL
S3160	Ethynodiol diacetate	77 mg/mL	77 mg/mL	<1 mg/mL

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Estrogen/progestogen Receptor

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Estrogen/progestogen Receptor Chemicals (24)water-soluble

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Estrogen/progestogen Receptor Chemicals (24)
water-soluble