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5-HT Receptor Antagonists and Agonists

  • Cat.No
  • Product Name
  • Information
  • Publications
  • Customer Reviews
  • S1243
  • Agomelatine
  • Agomelatine is classified as a norepinephrine-dopamine disinhibitor (NDDI) due to its antagonism of the 5-HT2C receptor.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2698
  • RS-127445
  • RS-127445 is a potent, selective and high affinity serotonin 5-HT2B receptor antagonist with a pIC50 of 10.4.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2663
  • WAY-100635
  • WAY-100635 is a potent and selective 5-hydroxytryptamine1A antagonist with an IC50 of 0.95 ± 0.12 nM for 5-HT
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S1615
  • Risperidone (Risperdal)
  • Risperidone(Risperdal) is an atypical antipsychotic used to treat schizophrenia.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2691
  • BMY 7378
  • BMY 7378 is a 5-HT1A receptor weak partial agonist/antagonist and α1D-adrenergic receptor antagonist with Ki values of 2.8 and 0.6 μM for cloned rat rat α1A and hamster α1B receptors, respectively.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2677
  • BRL-15572
  • BRL-15572 is a hydrochloride salt form of BRL-15572 which is a selective serotonin receptor subtype 5-HT1D antagonist with an IC50 of 260 μM.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2669
  • LY310762
  • LY310762 is a potent and selective 5-HT1D serotonin receptor antagonist with an EC50 of 31 nM.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)