Cyclobenzaprine HCl

Synonyms: Cyclobenzaprine hydrochloride

Cyclobenzaprine HCl(Cyclobenzaprine hydrochloride) is a muscle relaxant by blocking pain sensations, used for the treatment of muscle spasms; A 5-HT2 receptor antagonist.

Cyclobenzaprine HCl Chemical Structure

Cyclobenzaprine HCl Chemical Structure

CAS: 6202-23-9

Purity & Quality Control

Batch: S428301 DMSO] 62 mg/mL] false] Water] 62 mg/mL] false] Ethanol] 62 mg/mL] false Purity: 99.97%
99.97

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Biological Activity

Description Cyclobenzaprine HCl(Cyclobenzaprine hydrochloride) is a muscle relaxant by blocking pain sensations, used for the treatment of muscle spasms; A 5-HT2 receptor antagonist.
Targets
5-HT2 receptor [1]
NCT Number Recruitment Conditions Sponsor/Collaborators Start Date Phases
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NCT03443960 Completed
Healthy Subjects
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NCT03168022 Completed
Healthy Adults
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Lynn Henry|Damon Runyon Cancer Research Foundation|University of Michigan Rogel Cancer Center
August 2013 Phase 2

Chemical Information & Solubility

Molecular Weight 311.85 Formula

C20H22ClN

CAS No. 6202-23-9 SDF Download Cyclobenzaprine HCl SDF
Smiles CN(C)CCC=C1C2=CC=CC=C2C=CC3=CC=CC=C31.Cl
Storage (From the date of receipt)

In vitro
Batch:

DMSO : 62 mg/mL ( (198.81 mM); Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Water : 62 mg/mL

Ethanol : 62 mg/mL


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In vivo
Batch:

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In vivo Formulation Calculator

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In vivo Formulation Calculator (Clear solution)

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH2O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such
as vortex, ultrasound or hot water bath can be used to aid dissolving.

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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