GABA Receptor

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GABA Receptor Inhibitors | Activators | Agonists | Antagonists | Chemicals (14)

water-soluble

Cat.No. Product Name Information Product Use Citation Customer Product Validation
S1332 Flumazenil Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses.
S1338 Gabapentin HCl Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
S1329 Etomidate Etomidate is a GABAA receptor agonist, used as a short-acting anaesthetic agent or sedative.
S2133 Gabapentin Gabapentin is a GABA analogue, used to treat seizures and neuropathic pain.
S7071 (+)-Bicuculline (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.
  • Sci Rep, 2014, 4:7270
S1168 Valproic acid sodium salt (Sodium valproate) Valproic acid sodium salt (Sodium valproate) is a HDAC inhibitor by selectively inducing proteasomal degradation of HDAC2, used in the treatment of epilepsy, bipolar disorder and prevention of migraine headaches.
  • Nat Biotechnol, 2015, 10.1038/nbt.3130
  • J Neurosci, 2013, 33(17):7535-47
  • Cell Death Dis, 2016, 7:e2221
S1969 Nefiracetam Nefiracetam is a GABAergic, cholinergic, and monoaminergic neuronal system enhancer for Ro 5-4864-induced convulsions. Phase 2.
S3072 (R)-baclofen (R)-baclofen is a derivative of gamma-aminobutyric acid primarily used to treat spasticity.
S3018 Niflumic acid Niflumic acid is an inhibitor of cyclooxygenase-2 used for joint and muscular pain.
S2269 Baicalin Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors.
  • J Nutr Biochem, 2013, 24(11):1953-62
Cat.No. Product Name Information Product Use Citation Customer Product Validation
S2399 Dihydromyricetin Dihydromyricetin (Ampelopsin, Ampeloptin) is a natural antioxidant flavonoid from Ampelopsis grossedentata.
  • Food Chem Toxicol, 2012, 50(7):2508-14
S4197 Bemegride Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning.
S2026 Ginkgolide A Ginkgolide A is an extract from in Ginkgo biloba and a g-aminobutyric acid (GABA) antagonist with a Ki of 14.5 μM.
S4270 Oxiracetam Oxiracetam, a cyclic derivative of gamma-aminobutyric acid (GABA), is used as a nootropic drug to improve memory and learning.

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Cat.No. Product Name Solubility (25°C)
Water DMSO Ethanol
S1332 Flumazenil <1 mg/mL 5 mg/mL <1 mg/mL
S1338 Gabapentin HCl 42 mg/mL <1 mg/mL <1 mg/mL
S1329 Etomidate <1 mg/mL 49 mg/mL 49 mg/mL
S2133 Gabapentin 34 mg/mL <1 mg/mL <1 mg/mL
S7071 (+)-Bicuculline <1 mg/mL 21 mg/mL <1 mg/mL
S1168 Valproic acid sodium salt (Sodium valproate) 33 mg/mL 33 mg/mL 33 mg/mL
S1969 Nefiracetam 5 mg/mL 49 mg/mL 49 mg/mL
S3072 (R)-baclofen 8 mg/mL <1 mg/mL <1 mg/mL
S3018 Niflumic acid <1 mg/mL 56 mg/mL <1 mg/mL
S2269 Baicalin <1 mg/mL 89 mg/mL <1 mg/mL
S2399 Dihydromyricetin <1 mg/mL 64 mg/mL 64 mg/mL
S4197 Bemegride <1 mg/mL 31 mg/mL 31 mg/mL
S2026 Ginkgolide A <1 mg/mL 81 mg/mL 2 mg/mL
S4270 Oxiracetam 31 mg/mL 31 mg/mL <1 mg/mL
Tags: GABA inhibition | GABA receptor activation | GABA function | GABA drugs | GABA activity | GABA pathway | GABA-A receptor function | GABA receptor function | GABA activation | gamma aminobutyric acid function | GABA cancer | GABA assay | GABA receptor drugs | GABA receptor inhibition | GABA receptor signaling | GABA receptors review | GABA agonists list | GABA antagonist drugs | GABA inhibitor drugs | GABA inhibitor review
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