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S1250
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MDV3100 (Enzalutamide) |
MDV3100 is an androgen-receptor (AR) antagonist with IC50 of 36 nM. |
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S1190
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Bicalutamide (Casodex) |
Bicalutamide (Casodex, Cosudex, Calutide, Kalumid) is an androgen receptor (AR) antagonist with IC50 of 0.16 μM. |
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S1174
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Ostarine(MK-2866) |
Ostarine (GTx-024, MK-2866, Enobosarm, S-22) is a selective androgen receptor modulator (SARM) with Ki of 3.8 nM. |
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S1304
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Megestrol Acetate |
Megestrol Acetate is a synthetic progesteronal agent with an IC50 of 260 μM for the inhibition of HegG2. |
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S2042
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Cyproterone acetate |
Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM. |
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S4054
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Spironolactone |
Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM. |
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S2803
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Galeterone (TOK-001) |
Galeterone (TOK-001, VN/124-1) is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively. |
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S1140
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Andarine (GTX-007) |
Andarine (GTX-007) is a selective nonsteroidal androgen receptor (AR) agonist with Ki of 4 nM. |
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S2604
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Dehydroepiandrosterone(DHEA) |
Dehydroepiandrosterone(DHEA) is a 19-carbon endogenous natural steroid hormone. |
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