Research Area
Product Type
United States ( Change Country )
Bicalutamide (Casodex) Chemical Structure
Andarine (GTX-007)
Andarine (GTX-007) is an investigational selective androgen receptor modulator (SARM) and an active partial agonist.
Ostarine(MK-2866)
An androgen receptor modulator (SARM)
MDV3100 (Enzalutamide)
MDV3100 (Enzalutamide) is androgen-receptor inhibitor. Highly recommended inhibitor in AR research.
Synephrine (Oxedrine)
Synephrine (Oxedrine) is a compound commonly used for weight loss.
Andarine (GTX-007)
Andarine (GTX-007) is an investigational selective androgen receptor modulator (SARM) and an active partial agonist.
Ostarine(MK-2866)
An androgen receptor modulator (SARM)
Anastrozole
Anastrozole inhibits the enzyme aromatase.
Fulvestrant (Faslodex)
Fulvestrant (Faslodex) is a Synthetic estrogen receptor antagonist(SERD)
Exemestane
Exemestane was found to inhibit human placental aromatase with IC50 of 42 nM.
Finasteride
Finasteride is an inhibitor of steroid Type II 5α-reductase.
Biological Activity
Bicalutamide (Casodex) is an active competitive non-steroidal androgen receptor antagonist. Bicalutamide (Casodex) is an oral non-steroidal anti-androgen used in the treatment of prostate cancer and hirsutism. Bicalutamide (Casodex)belongs to a class of agents called anti-androgens which includes flutamide (Eulexin) and nilutamide (Nilandron). Bicalutamide (Casodex)acts as a pure anti-androgen by binding to the androgen receptor (AR) and preventing the activation of the AR and subsequent upregulation of androgen responsive genes by androgenic hormones. In addition, bicalutamide (Casodex, Cosudex, Calutide, Kalumid) accelerates the degradation of the androgen receptor. [1][2]
References on Bicalutamide (Casodex)
- [] BIOPHARMACEUTICS & DRUG DISPOSITION 1997;18:6, 499±507
Product Information
| Molecular Weight (WM): | 430.37 |
|---|---|
| Formula: | C18H14F4N2O4S |
| CAS No.: | 90357-06-5 |
| Synonyms: |
N/A
|
| Dissolve in (25°C): | DMSO ≥86mg/mL |
| Water <1mg/mL | |
| Ethanol ≥7mg/mL | |
| Storage: | 2 years-20°CPowder |
| 1 week-4°Cin DMSO | |
| 1 month-80°in DMSO |
Quality Control & MSDS
Research Area
Related Inhibitors
Recommended Screening Libraries
Chemical Library
A collection of 864 bioactive compounds
Inhibitor Library
A collection of 481 inhibitors
Kinase Inhibitor Library
A collection of 194 kinase inhibitors
Tyrosine Kinase Inhibitor Library
A collection of 85 tyrosine kinase inhibitors.
FDA Approved Drug Library
A collection of 426 FDA approved drugs
Natural Product Library
A collection of 139 natural products
Chemotherapeutic Agent Library
A collection of 40 chemotherapeutic agents
Epigenetics Compound library
A unique collection of 17 small molecule modulators
Stem Cell Compound library
A unique collection of 47 small molecule inhibitors
GPCR Compound library
A unique collection of 63 GPCR small molecules
Keywords:buy Bicalutamide (Casodex) | Bicalutamide (Casodex) supplier | purchase Bicalutamide (Casodex) | Bicalutamide (Casodex) cost | Bicalutamide (Casodex) manufacturer | order Bicalutamide (Casodex) | Bicalutamide (Casodex) distributor