GluR Glutamate Receptor

Cat.No.	Product Name	Information	Product Citations
S2251	(-)-Huperzine A	(-)-Huperzine A is a potent, highly specific and reversible inhibitor of acetylcholinesterase (AChE) with K_i of 7 nM.
S2857	Dizocilpine (MK 801)	Dizocilpine is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with K_i of 30.5 nM.
S6001	LY2140023 (LY404039)	LY404039 is a potent agonist of recombinant human mGlu2, mGlu3 receptors and rat neurons expressing native mGlu2/3 receptors with K_i of 149 nM, 92 nM and 88 nM, respectively.	Neuropharm, 2012, 62(7), 2184-2191 PLoS One, 2011, 6(7):e22235 Synapse, 2009, 63(10), 935-939
S1245	Dimebon (Latrepirdine)	Dimebon is an antihistamine drug.
S2690	ADX-47273	ADX47273 is a potent and specific mGlu5 antagonist with IC50 of 0.17μM.
S7072	NMDA (N-Methyl-D-aspartic acid)	NMDA（N-Methyl-D-aspartic acid）is a specific agonist for NMDA receptor mimicking the action of L-glutamate receptor.
S2795	VU 0357121	VU0357121 is a novel allosteric modulator of mGlu5 with EC50 of 33 nM.
S2809	MPEP	MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM.
S2861	CTEP	CTEP is a selective allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM.
S2876	(-)-MK 801 Maleate	MK-801 is a potent, selective and non-competitive NMDA receptor antagonist with K_d of 37.2 nM in rat brain membranes.

Cat.No.	Product Name	Information	Product Citations	Customer Reviews
S2862	VU 0364770	VU 0364770 is a selective positive allosteric mGlu4 with EC50 of 1.1 μM.
S2892	VU 0361737	VU 0361737 is a selective positive allosteric modulator for mGlu4 receptor with EC50 of 240 nM and 110 nM at human and rat receptors, respectively.

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