Glucocorticoid Receptor

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S1707 Eplerenone <1 mg/mL 4 mg/mL <1 mg/mL
S1696 Hydrocortisone <1 mg/mL 73 mg/mL 23 mg/mL
S1737 Prednisolone <1 mg/mL 72 mg/mL 10 mg/mL
S1622 Prednisone <1 mg/mL 71 mg/mL <1 mg/mL
S1669 Loteprednol etabonate <1 mg/mL 93 mg/mL 4 mg/mL
S5685 Desoximetasone <1 mg/mL 75 mg/mL 75 mg/mL
S5486 Fluorometholone <1 mg/mL 75 mg/mL 5 mg/mL
S4775 Cortodoxone -1 mg/mL 69 mg/mL -1 mg/mL
S1987 Mometasone furoate <1 mg/mL 6 mg/mL <1 mg/mL
S1992 Fluticasone propionate <1 mg/mL 100 mg/mL 5 mg/mL
S1733 Methylprednisolone <1 mg/mL 75 mg/mL 2 mg/mL
S1286 Budesonide <1 mg/mL 86 mg/mL 19 mg/mL
S1628 Triamcinolone Acetonide <1 mg/mL 87 mg/mL 13 mg/mL
S1689 Meprednisone <1 mg/mL 75 mg/mL 4 mg/mL
S1888 Deflazacort <1 mg/mL 88 mg/mL 12 mg/mL
S2470 Fluocinolone Acetonide <1 mg/mL 90 mg/mL 12 mg/mL
S1688 Betamethasone Dipropionate <1 mg/mL 100 mg/mL 66 mg/mL
S1690 Betamethasone Valerate <1 mg/mL 95 mg/mL 58 mg/mL
S2570 Prednisolone Acetate <1 mg/mL 81 mg/mL <1 mg/mL
S1500 Betamethasone <1 mg/mL 79 mg/mL 10 mg/mL
S4088 Flumethasone <1 mg/mL 82 mg/mL 6 mg/mL
S1701 Desonide <1 mg/mL 83 mg/mL 30 mg/mL
S2608 Fluocinonide <1 mg/mL 99 mg/mL <1 mg/mL
S2584 Clobetasol propionate <1 mg/mL 93 mg/mL 20 mg/mL
S1933 Triamcinolone <1 mg/mL 78 mg/mL 1 mg/mL
S3078 Beclomethasone dipropionate <1 mg/mL 104 mg/mL 18 mg/mL
S2559 Cortisone acetate <1 mg/mL 7 mg/mL <1 mg/mL
S3617 (20S)-Protopanaxatriol <1 mg/mL 95 mg/mL 95 mg/mL
S4752 Corticosterone <1 mg/mL 69 mg/mL 69 mg/mL
S4228 Fluorometholone Acetate <1 mg/mL 83 mg/mL 1 mg/mL
Catalog No. Information Product Use Citations Product Validations
S1707

Eplerenone

Eplerenone is a mineralocorticoid receptor antagonist, and blocks the action of aldosterone, used to control high blood pressure.
S1696

Hydrocortisone

Hydrocortisone is a steroid hormone or glucocorticoid produced by the adrenal gland.
S1737

Prednisolone

Prednisolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
J Pharmacol Exp Ther, 2014, 350(3):646-56
PLoS One, 2014, 9(12):e111840
Leuk Lymphoma, 2014, 55(5):1144-50
S1622

Prednisone

Prednisone (Adasone) is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound.
S1669

Loteprednol etabonate

Loteprednol etabonate is a potent glucocorticoid receptor agonist, used in treatment of inflammation of the eye due to allergies.
S5685New

Desoximetasone

Desoximetasone is a synthetic glucocorticoid receptor agonist with metabolic, anti-inflammatory and immunosuppressive activity.
S5486New

Fluorometholone

Fluorometholone is a synthetic glucocorticoid with anti-inflammatory and anti-allergic properties. It is usually used as eye drops in the treatment of allergic and inflammatory conditions of the eye.
S4775New

Cortodoxone

Cortodoxone, also known as 11-Deoxycortisol, is a glucocorticoid steroid hormone.
S1987

Mometasone furoate

Mometasone Furoate is a glucocorticoid receptor agonist, used topically to reduce inflammation of the skin or in the airways.
S1992

Fluticasone propionate

Fluticasone Propionate is a synthetic glucocorticoid, used to treat non-allergic and allergic rhinitis.
S1733

Methylprednisolone

Methylprednisolone is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation.
Trop J Pharm Res, 2014, 13 (1): 53-59
S1286

Budesonide

Budesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis.
S1628

Triamcinolone Acetonide

Triamcinolone acetonide is a synthetic glucocorticoid, used in the symptomatic treatment of inflammation.
S1689

Meprednisone

Meprednisone is a glucocorticoid and a methylated derivative of prednisone.
S1888

Deflazacort

Deflazacort is a glucocorticoid used as an anti-inflammatory and immunosuppressant.
S2470

Fluocinolone Acetonide

Fluocinolone Acetonide is a corticosteroid that binds to the cytosolic glucocorticoid receptor.
S1688

Betamethasone Dipropionate

Betamethasone Dipropionate is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities.
S1690

Betamethasone Valerate

Betamethasone Valerate is a moderately potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.
S2570

Prednisolone Acetate

Prednisolone Acetate is a synthetic corticosteroid drug that is particularly effective as an immunosuppressant agent.
S1500

Betamethasone

Betamethasone is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.
S4088

Flumethasone

Flumethasone is a glucocorticoid receptor agonist, this complex binds to the nucleus causing a variety of genetic activation and repressions.
S1701

Desonide

Desonide is a low potency topical corticosteroid.
S2608

Fluocinonide

Fluocinonide (Vanos) is a potent glucocorticoid steroid used topically as anti-inflammatory agent for the treatment of skin disorders such as eczema.
S2584

Clobetasol propionate

Clobetasol propionate is an anti-inflammatory corticosteroid used to treat various skin disorders.
S1933

Triamcinolone

Triamcinolone is a glucocorticoid given, as the free alcohol or in esterified form, orally, intramuscularly, by local injection, by inhalation, or applied topically in the management of various disorders in which corticosteroids are indicated.
S3078

Beclomethasone dipropionate

Beclomethasone dipropionate is a potent glucocorticoid steroid used for the treatment of rhinitis and sinusitis.
S2559

Cortisone acetate

Cortisone acetate (Cortone) is an acetate salt form of cortisone that is a steroid hormone and a glucocorticoid.
S3617

(20S)-Protopanaxatriol

(20S)-Protopanaxatriol(g-PPT), a neuroprotective metabolite of ginsenoside, protopanaxatriol (g-PPT), is a functional ligand for both GR and ERbeta and could modulate endothelial cell functions through the glucocorticoid receptor (GR) and oestrogen receptor (ER).

S4752

Corticosterone

Corticosterone, the major stress hormone, is an adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid.
Xenobiotica, 2016, 46(10):948-52
S4228

Fluorometholone Acetate

Fluorometholone Acetate is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.