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Glucocorticoid Receptor

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Cat.No. Product Name Information Product Use Citations Product Validations
E1091 Relacorilant (CORT125134) Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.
Biomed Pharmacother, 2024, 180:117523
Journal of Endocrinological Investigation, 2023, 1-14
J Endocrinol Invest, 2023, 10.1007/s40618-023-02184-3
S1322 Dexamethasone Dexamethasone is a potent synthetic member of the glucocorticoid class of steroid drugs, and an interleukin receptor modulator that has anti-inflammatory and immunosuppressant effects. Dexamethasone induces autophagy and mitophagy. Dexamethasone is tested in hospitalized patients with COVID-19 and is found to have benefits for critically ill patients.
Signal Transduct Target Ther, 2025, 10(1):230
Signal Transduct Target Ther, 2025, 10(1):394
Gut, 2025, gutjnl-2025-336105
Verified customer review of Dexamethasone
S1696 Hydrocortisone (Cortisol) Hydrocortisone is a steroid hormone or glucocorticoid produced by the adrenal gland.
Bone Res, 2025, 13(1):37
Clin Cancer Res, 2025, 10.1158/1078-0432.CCR-24-1812
Cell Death Discov, 2025, 11(1):286
S1737 Prednisolone Prednisolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. This compound is widely used in the treatment of various inflammatory and autoimmune conditions. It works by suppressing the immune response and reducing inflammation in the body. The efficacy of this medication has been well-documented in clinical studies. Patients prescribed this drug should follow their healthcare provider's instructions carefully to minimize potential side effects.
Cancers (Basel), 2025, 17(12)2034
Front Oncol, 2025, 15:1520972
Molecules, 2024, 29(7)1546
Verified customer review of Prednisolone
S5956 Dexamethasone phosphate disodium Dexamethasone phosphate disodium is a glucocorticoid receptor agonist with both anti-inflammatory and anti-oxidative effects.
Cell Rep Med, 2025, S2666-3791(25)00102-8
Cell Rep, 2023, 42(6):112566
Blood Adv, 2023, 7(4):469-481
S4646 Ciclesonide Ciclesonide (Alvesco, Omnaris, RPR251526, Zetonna) is a glucocorticoid used to treat obstructive airway diseases.
Proceedings of the National Academy of Sciences, November 2025, 122(48)
American Journal of Physiology-Lung Cellular and Molecular Physiology, May 1, 2023, L722-L736
American Journal of Physiology-Lung Cellular and Molecular Physiology, May 1, 2023, L722-L736
S1622 Prednisone Prednisone is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound.
Bangladesh Journal of Pharmacology, December 13, 2024, 73-80
Frontiers in Immunology, August 13, 2021, 739605
PLoS One, August 1, 2018, e0200725
S2559 Cortisone acetate Cortisone acetate (Cortone, NSC 49420) is an acetate salt form of cortisone that is a steroid hormone and a glucocorticoid.
Cancer Immunology, Immunotherapy, 2025, 316
Cancer Immunol Immunother, 2025, 74(10):316
iScience, 2024, 27(10):110862
S1286 Budesonide Budesonide(Labazenit) is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis.
Arch Toxicol, 2025, 99(3):1105-1116
bioRxiv, 2025, 2025.03.31.646052
Front Mol Neurosci, 2024, 17:1473960
S1628 Triamcinolone Acetonide Triamcinolone acetonide is a synthetic glucocorticoid, used in the symptomatic treatment of inflammation. This compound is a synthetic glucocorticoid, used in the symptomatic treatment of inflammation.
Arch Toxicol, 2025, 99(3):1105-1116
FASEB J, 2025, 39(1):e70298
The FASEB Journal, 2025, e70298