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Progesterone Receptor

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Cat.No. Product Name Information Product Use Citations Product Validations
S2567 Medroxyprogesterone Acetate (MPA) MPA (Medroxyprogesterone acetate) is a synthetic progestin and act as a potent progesterone receptor agonist, used to treat abnormal menstruation or irregular vaginal bleeding.
Cancer Sci, 2025, 10.1111/cas.70081
Cell Prolif, 2024, e13780.
J Transl Med, 2024, 22(1):478
Verified customer review of Medroxyprogesterone Acetate (MPA)
S4040 Norethindrone Norethindrone (Norethisterone) is a synthetic progestin, which mimic the actions of the endogenous ovarian hormone progesterone.
Nature Cancer, 2020, 235-248
Nat Cancer, 2020, 1(2):235-248
S2606 Mifepristone (RU-486) Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. Mifepristone promotes cell autophagy and apoptosis, decreases Bcl-2 level and increases Beclin1 level, accompanied by weakened interaction between Bcl-2 and Beclin1.Mifepristone (RU486) can be used to induce animal models of Spontaneous Abortion.
Alcoholism: Clinical and Experimental Research, May 2020, 1025-1036
Scientific Reports, March 24, 2020, 5363
Frontiers in Immunology, August 12, 2022, 863034
Verified customer review of Mifepristone (RU-486)
S1705 Progesterone Progesterone is an endogenous steroid hormone involved in the menstrual cycle, pregnancy, and embryogenesis of humans and other species. This compound is a potent agonist of the nuclear progesterone receptor (nPR) with Kd of 1 nM; an agonist of the membrane progesterone receptors(mPRs); an antagonist of the σ1 receptor.
Bone Res, 2025, 13(1):37
Cell Proliferation, 2025, e70025
Nat Commun, 2024, 15(1):8708
Verified customer review of Progesterone
S1304 Megestrol Acetate Megestrol acetate (BDH1298, SC10363) is a synthetic progestogen, used to treat breast cancer and loss of appetite.
Scientific Reports, October 06, 2017, 12754
OncoTargets and Therapy, October 03, 2017, 4809-4819
iScience, 2024, 27(10):110862
Verified customer review of Megestrol Acetate
S1377 Drospirenone Drospirenone (ZK 3059) is a synthetic progestin that is an analog to spironolactone.
Acta Pharmaceutica Sinica B, 2023, 662-677
Acta Pharm Sin B, 2023, 13(2):662-677
Nature Cancer, 2020, 235-248
S3081 Ulipristal Acetate (CDB 2914) Ulipristal acetate (CDB-2914, HRP 2000, RU 44675) is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.
Nature, 2025, 10.1038/s41586-025-09684-7
The Journal of Clinical Endocrinology & Metabolism, 2019, 6256–6264
J Clin Endocrinol Metab, 2019, 104(12):6256-6264
S3635 Medroxyprogesterone Medroxyprogesterone (MP) is a synthetic pregnane steroid and a derivative of progesterone. It is a potent progesterone receptor agonist.
Theranostics, 2024, 593-607
S1251 Dienogest Dienogest (STS 557) is an orally active synthetic progesterone, used for contraception and the treatment of endometriosis.
S3167 Altrenogest Altrenogest (A35957, RU2267,R2267) is a progestogen structurally related to veterinary steroid trenbolone.