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Progesterone Receptor

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Cat.No. Product Name Information Product Use Citations Product Validations
S4040 Norethindrone Norethindrone (Norethisterone) is a synthetic progestin, which mimic the actions of the endogenous ovarian hormone progesterone.
Nat Cancer, 2020, 1(2):235-248
S2606 Mifepristone (RU-486) Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. Mifepristone promotes cell autophagy and apoptosis, decreases Bcl-2 level and increases Beclin1 level, accompanied by weakened interaction between Bcl-2 and Beclin1.Mifepristone (RU486) can be used to induce animal models of Spontaneous Abortion.
Pharmacol Res, 2025, 215:107696
Cell Death Dis, 2025, 16(1):237
J Virol, 2025, 99(2):e0147224
Verified customer review of Mifepristone (RU-486)
S2567 MPA (Medroxyprogesterone acetate) Medroxyprogesterone acetate (MPA) is a synthetic progestin that acts as a potent progesterone receptor agonist, used to treat abnormal menstruation or irregular vaginal bleeding.
Cancer Sci, 2025, 10.1111/cas.70081
Cell Prolif, 2024, e13780.
J Transl Med, 2024, 22(1):478
Verified customer review of MPA (Medroxyprogesterone acetate)
S1705 Progesterone Progesterone is an endogenous steroid hormone involved in the menstrual cycle, pregnancy, and embryogenesis of humans and other species. This compound is a potent agonist of the nuclear progesterone receptor (nPR) with Kd of 1 nM; an agonist of the membrane progesterone receptors(mPRs); an antagonist of the σ1 receptor.
Bone Res, 2025, 13(1):37
Nat Commun, 2024, 15(1):8708
Dev Cell, 2024, S1534-5807(24)00326-5
Verified customer review of Progesterone
S1304 Megestrol Acetate Megestrol acetate (BDH1298, SC10363) is a synthetic progestogen, used to treat breast cancer and loss of appetite.
iScience, 2024, 27(10):110862
J Pers Med, 2022, 12(2)258
Hum Cell, 2022, 10.1007/s13577-022-00671-y
Verified customer review of Megestrol Acetate
S1377 Drospirenone Drospirenone (ZK 3059) is a synthetic progestin that is an analog to spironolactone.
Acta Pharm Sin B, 2023, 13(2):662-677
Nat Cancer, 2020, 1(2):235-248
J Thromb Haemost, 2015, 13(10):1918-24
S3081 Ulipristal Acetate (CDB 2914) Ulipristal acetate (CDB-2914, HRP 2000, RU 44675) is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.
Nature, 2025, 10.1038/s41586-025-09684-7
J Clin Endocrinol Metab, 2019, 104(12):6256-6264
Cell Prolif, 2017, 50(5)
S1251 Dienogest Dienogest (STS 557) is an orally active synthetic progesterone, used for contraception and the treatment of endometriosis.
S3167 Altrenogest Altrenogest (A35957, RU2267,R2267) is a progestogen structurally related to veterinary steroid trenbolone.
E0527 Norgestimate Norgestimate, a synthetic progesterone analog, is an orally active progestin with highly selective progestational activity and minimal androgenicity.