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S1076
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SB 203580 |
SB203580 is a p38 MAPK inhibitor with IC50 of 0.3-0.5 μM and blocks PKB phosphorylation with IC50 of 3-5 μM. |
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S1574
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BIRB 796 (Doramapimod) |
BIRB 796 (Doramapimod) is a highly selective p38α MAPK inhibitor with Kd of 0.1 nM. |
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S1077
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SB 202190 |
SB 202190 (FHPI) is a potent p38 MAPK inhibitor targeting p38α and p38β with IC50 of 50 nM and 100 nM, respectively. |
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S1494
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LY2228820 |
LY2228820 is a novel and potent inhibitor of p38 MAPK with IC50 of 7 nM. |
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S6005
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VX-702 |
VX-702 is a highly selective inhibitor of p38 MAPKα with IC50 of 4-20 nM. |
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S1527
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Vinorelbine (Navelbine) |
Vinorelbine (Navelbine) is an anti-mitotic agent which inhibits the proliferation of Hela cells with IC50 of 1.25 nM. |
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S2726
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PH-797804 |
PH-797804 is a novel pyridinone inhibitor of p38α with IC50 of 26 nM. |
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S1458
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VX-745 |
VX-745 is a potent and selective inhibitor of p38α MAPK and p38β MAPK with IC50 of 10 nM and 220 nM, respectively. |
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S2928
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TAK 715 |
TAK 715 is a p38 MAPK inhibitor for p38α with IC50 of 7.1 nM. |
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