HIV Protease

Sigaling Pathway Map

Research Area

  • Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S1185 Ritonavir <1 mg/mL 100 mg/mL 3 mg/mL
S1380 Lopinavir <1 mg/mL 126 mg/mL 126 mg/mL
S1457 Atazanavir Sulfate <1 mg/mL 104 mg/mL <1 mg/mL
S1620 Darunavir Ethanolate <1 mg/mL 100 mg/mL <1 mg/mL
S1639 Amprenavir <1 mg/mL 16 mg/mL 100 mg/mL
S4662 Atazanavir <1 mg/mL 100 mg/mL 32 mg/mL
S2319 Limonin <1 mg/mL 44 mg/mL <1 mg/mL
S4282 Nelfinavir Mesylate <1 mg/mL 100 mg/mL 100 mg/mL
S7381 Pepstatin A <1 mg/mL 100 mg/mL 1 mg/mL
Catalog No. Information Product Use Citations Product Validations
S1185

Ritonavir

Ritonavir is a Cytochrome P450 3A and Protease Inhibitor; Also inhibits Cytochrome P450 2D6, P-Glycoprotein and induces Cytochrome P450 2C19, Cytochrome P450 1A2, Cytochrome P450 2C9, Cytochrome P450 2B6 and UDP Glucuronosyltransferases.

S1380

Lopinavir

Lopinavir is a potent HIV protease inhibitor with Ki of 1.3 pM in a cell-free assay.

S1457

Atazanavir Sulfate

Atazanavir Sulfate is a HIV protease inhibitor with Ki of 2.66 nM in a cell-free assay.

S1620

Darunavir Ethanolate

Darunavir Ethanolate (DRV) is a nonpeptidic HIV protease inhibitor, used to treat HIV infection.

S1639

Amprenavir

Amprenavir is a potent PXR-selective agonist, and an HIV protease inhibitor, used to treat HIV.

S4662New

Atazanavir

Atazanavir is an azapeptide and HIV-protease inhibitor that is used in the treatment of HIV infections and AIDS in combination with other anti-HIV agents.

S2319

Limonin

Limonin is a triterpenoid enriched in citrus fruits, which has antivirus and antitumor ability.

S4282

Nelfinavir Mesylate

Nelfinavir Mesylate is a potent HIV protease inhibitor with Ki of 2 nM.

S7381

Pepstatin A

Pepstatin A is a potent aspartic protease inhibitor, and also inhibits HIV replication.

Catalog No. Information Product Use Citations Product Validations
S1185

Ritonavir

Ritonavir is a Cytochrome P450 3A and Protease Inhibitor; Also inhibits Cytochrome P450 2D6, P-Glycoprotein and induces Cytochrome P450 2C19, Cytochrome P450 1A2, Cytochrome P450 2C9, Cytochrome P450 2B6 and UDP Glucuronosyltransferases.

S1380

Lopinavir

Lopinavir is a potent HIV protease inhibitor with Ki of 1.3 pM in a cell-free assay.

S1457

Atazanavir Sulfate

Atazanavir Sulfate is a HIV protease inhibitor with Ki of 2.66 nM in a cell-free assay.

S1620

Darunavir Ethanolate

Darunavir Ethanolate (DRV) is a nonpeptidic HIV protease inhibitor, used to treat HIV infection.

S1639

Amprenavir

Amprenavir is a potent PXR-selective agonist, and an HIV protease inhibitor, used to treat HIV.

S4662New

Atazanavir

Atazanavir is an azapeptide and HIV-protease inhibitor that is used in the treatment of HIV infections and AIDS in combination with other anti-HIV agents.

S2319

Limonin

Limonin is a triterpenoid enriched in citrus fruits, which has antivirus and antitumor ability.

S4282

Nelfinavir Mesylate

Nelfinavir Mesylate is a potent HIV protease inhibitor with Ki of 2 nM.

S7381

Pepstatin A

Pepstatin A is a potent aspartic protease inhibitor, and also inhibits HIV replication.