AhR

Inhibitory Selectivity

AhR Products

New AhR Products
Catalog No. Information Product Use Citations Product Validations
S8842New

BAY-218

BAY-218 is a potent and selective small-molecule AhR inhibitor, inhibiting AhR nuclear translocation, dioxin response element (DRE)-luciferase reporter expression and AhR-regulated target gene expression induced by both exogenous and endogenous AhR ligands.

S2858

StemRegenin 1 (SR1)

StemRegenin 1 is an aryl hydrocarbon receptor (AhR) inhibitor with IC50 of 127 nM in a cell-free assay.

S7711

CH-223191

CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist with IC50 of 30 nM.

S6560New

PDM2

PDM2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.

s9092

Norisoboldine

Norisoboldine, a natural aryl hydrocarbon receptor (AhR) agonist, attenuates ulcerative colitis (UC) and induces the generation of Treg cells.

S7510

UM729

UM729 is an enhancer of aryl hydrocarbon receptor (AhR) antagonists.

Catalog No. Information Product Use Citations Product Validations
S8842New

BAY-218

BAY-218 is a potent and selective small-molecule AhR inhibitor, inhibiting AhR nuclear translocation, dioxin response element (DRE)-luciferase reporter expression and AhR-regulated target gene expression induced by both exogenous and endogenous AhR ligands.

Catalog No. Information Product Use Citations Product Validations
S2858

StemRegenin 1 (SR1)

StemRegenin 1 is an aryl hydrocarbon receptor (AhR) inhibitor with IC50 of 127 nM in a cell-free assay.

S7711

CH-223191

CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist with IC50 of 30 nM.

S6560New

PDM2

PDM2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.

Catalog No. Information Product Use Citations Product Validations
s9092

Norisoboldine

Norisoboldine, a natural aryl hydrocarbon receptor (AhR) agonist, attenuates ulcerative colitis (UC) and induces the generation of Treg cells.

Catalog No. Information Product Use Citations Product Validations
S7510

UM729

UM729 is an enhancer of aryl hydrocarbon receptor (AhR) antagonists.