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S2797
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Lonafarnib (SCH66336) |
Lonafarnib (SCH 66336) is a selectively FPTase inhibitor for H-ras, K-ras-4B and N-ras with IC50 of 1.9 nM, 5.2 nM and 2.8 nM, respectively. |
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S1453
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Tipifarnib (Zarnestra) |
Tipifarnib (Zarnestra, R115777) is a potent and specific farnesyltransferase (FTase) inhibitor with IC50 of 0.6 nM. |
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S2674
|
A 922500 |
A 922500 is a DGAT-1 inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively. |
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S2821
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RG108 |
RG108 is an inhibitor of DNA methyltransferase with IC50 of 115 nM. |
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S8006
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BIX01294 |
BIX01294 is an inhitor of G9a histone methyltransferase with IC50 of 2.7 μM. |
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S4021
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Tolcapone |
Tolcapone is a selective, potent and reversible of catechol-O-methyl transferase (COMT) inhibitor with Ki of 30 nM. |
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