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S2480
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Loperamide HCl |
Loperamide is an opioid-receptor agonist with an ED50 of 0.15 mg/kg. |
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S2722
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JTC-801 |
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM. |
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S1139
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ADL5859 HCl |
ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM. |
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S2503
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Racecadotril (Acetorphan) |
Racecadotril is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM |
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S2085
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Trimebutine |
Trimebutine is an agonist of peripheral mu, kappa and delta opiate receptors, used as spasmolytic agent for treatment of both acute and chronic abdominal pain.
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S1941
|
Enalapril maleate (Vasotec) |
Enalapril maleate (Vasotec), the active metabolite of enalapril, competes with angiotensin I for binding at the angiotensin-converting enzyme, blocking the conversion of angiotensin I to angiotensin II. |
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S2103
|
Naltrexone HCl |
Naltrexone is an opioid receptor antagonist with IC50 of 8 nM used primarily in the management of alcohol dependence and opioid dependence.
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S3066
|
Naloxone HCl |
Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose. |
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