Rucaparib Camsylate

For research use only.

Catalog No.S5195 Synonyms: Rubraca, AG014699 Camsylate, PF01367338 Camsylate

5 publications

Rucaparib Camsylate Chemical Structure

CAS No. 1859053-21-6

Rucaparib (Rubraca, AG014699, PF01367338) Camsylate is an inhibitor of PARP with Ki of 1.4 nM for PARP1 in a cell-free assay, also showing binding affinity to eight other PARP domains.

Selleck's Rucaparib Camsylate has been cited by 5 publications

Purity & Quality Control

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Biological Activity

Description Rucaparib (Rubraca, AG014699, PF01367338) Camsylate is an inhibitor of PARP with Ki of 1.4 nM for PARP1 in a cell-free assay, also showing binding affinity to eight other PARP domains.
Targets
PARP1 [1]
(Cell-free assay)
1.4 nM(Ki)

Protocol

Solubility (25°C)

In vitro DMSO 100 mg/mL (179.96 mM)
Water Insoluble
Ethanol Insoluble

* Please note that Selleck tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Chemical Information

Molecular Weight 555.66
Formula

C29H34FN3O5S

CAS No. 1859053-21-6
Storage powder
in solvent
Synonyms Rubraca, AG014699 Camsylate, PF01367338 Camsylate

In vivo Formulation Calculator (Clear solution)

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Molarity Calculator

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*When preparing stock solutions, please always use the batch-specific molecular weight of the product found on the via label and SDS / COA (available on product pages).

Dilution Calculator

Dilution Calculator

Calculate the dilution required to prepare a stock solution. The Selleck dilution calculator is based on the following equation:

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* When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / COA (available online).

The Serial Dilution Calculator Equation

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Mass Concentration Volume Molecular Weight

Clinical Trial Information

NCT Number Recruitment interventions Conditions Sponsor/Collaborators Start Date Phases
NCT01009190 Completed Drug: PF-01367338|Drug: Carboplatin Advanced Solid Tumors Clovis Oncology Inc. February 2010 Phase 1

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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PARP Signaling Pathway Map

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Cell Lines Assay Type Concentration Incubation Time Formulation Activity Description PMID