κ-opioid receptor Selective Agonists
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
Matrine((+)-Matrine) is an alkaloid found in plants from the Sophora family, which has a variety of pharmacological effects, including anti-cancer effects, and action as a kappa opioid receptor agonist.
ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel. Phase 2.
|Pan||κ-opioid receptor, Ki: 37 nM|