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S3021
|
Rimonabant (SR141716) |
Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane. |
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S1544
|
AM-1241 |
AM-1241 is a selective CB2 agonist with Ki of 3.4 nM. |
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S2819
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AM251 |
AM251 is a cannabinoid 1 receptor antagonist with IC50 of 8.9 μM. |
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S1534
|
Org 27569 |
Org 27569 is an allosteric modulator of CB1 cannabinoid receptor. |
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S2778
|
GW842166X |
GW842166X is a potent and highly selective agonist of CB2 receptor. |
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S2854
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BML-190 |
BML-190 is a selective CB2 inverse agonist with Ki of 435 nM. |
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S8012
|
Otenabant (CP-945598) HCl |
CP-945598 HCl is a potent and selective cannabinoid type 1 receptor antagonist with Ki of 0.7 nM. |
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