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United States ( Change Country )
Org 27569 Chemical Structure
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Biological Activity
Org 27569 is an allosteric modulator of CB1 cannabinoid receptor. It significantly increases the binding of CB1 receptor agonist [3H]-CP 55,940 (pKB = 5.67) and causes a significant decrease in specific binding of CB1 receptor inverse agonist SR141716A (Rimonabant; pKB = 5.95); in the reporter gene assay behaves as insurmountable CP 55,940 antagonist; pKB = 7.57 at CB1 receptors in mouse vas deferens. [1][2]
Chemical Information
| Molecular Weight (WM): | 409.95 |
|---|---|
| Formula: | C24H28ClN3O |
| CAS No.: | 868273-06-7 |
| Synonyms: |
Org27569
|
| Dissolve in (25°C): | |
| Storage: | 2 years-20°CPowder |
| 1 week-4°Cin DMSO | |
| 1 month-80°in DMSO |
Quality Control & MSDS
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