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Cannabinoid Receptor

Compare Cannabinoid Receptor Chemicals

Compare Cannabinoid Receptor Inhibitors

Inhibitory Selectivity
Solubility

Cat.No.	Product Name	Solubility (25°C)
Cat.No.	Product Name	Water	DMSO	Ethanol
S3021	Rimonabant (SR141716)	<1 mg/mL	25 mg/mL	2 mg/mL
S1544	AM-1241	<1 mg/mL	101 mg/mL	<1 mg/mL
S2819	AM251	<1 mg/mL	40 mg/mL	<1 mg/mL
S2778	GW842166X	<1 mg/mL	20 mg/mL	<1 mg/mL
S2854	BML-190	<1 mg/mL	22 mg/mL	<1 mg/mL
S8012	Otenabant (CP-945598) HCl	<1 mg/mL	1(加热) mg/mL	<1 mg/mL

Research Area
Research Area

Cannabinoid Receptor Chemicals (7)
water-soluble

Cat.No.	Product Name	Information	Product Citations	Customer Reviews
S3021	Rimonabant (SR141716)	Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
S1544	AM-1241	AM-1241 is a selective CB2 agonist with K_i of 3.4 nM.
S2819	AM251	AM251 is a cannabinoid 1 receptor antagonist with IC50 of 8.9 μM.
S1534	Org 27569	Org 27569 is an allosteric modulator of CB1 cannabinoid receptor.
S2778	GW842166X	GW842166X is a potent and highly selective agonist of CB2 receptor.
S2854	BML-190	BML-190 is a selective CB2 inverse agonist with K_i of 435 nM.
S8012	Otenabant (CP-945598) HCl	CP-945598 HCl is a potent and selective cannabinoid type 1 receptor antagonist with K_i of 0.7 nM.

Inhibitory Selectivity
Solubility

Cat.No.	Product Name	Solubility (25°C)
Cat.No.	Product Name	Water	DMSO	Ethanol
S3021	Rimonabant (SR141716)	<1 mg/mL	25 mg/mL	2 mg/mL
S1544	AM-1241	<1 mg/mL	101 mg/mL	<1 mg/mL
S2819	AM251	<1 mg/mL	40 mg/mL	<1 mg/mL
S2778	GW842166X	<1 mg/mL	20 mg/mL	<1 mg/mL
S2854	BML-190	<1 mg/mL	22 mg/mL	<1 mg/mL
S8012	Otenabant (CP-945598) HCl	<1 mg/mL	1(加热) mg/mL	<1 mg/mL

Tags: Cannabinoid Receptor signaling | CB1 receptor signaling | CB2 signaling | Cannabinoid Receptor inhibitor review