CYP2 Selective Inhibitors
|Catalog No.||Product Name||Information||Selective / Pan||IC50 / Ki|
Benzbromarone is a CYP2C9 inhibitor, it binds to CYP2C9 with Ki value of 19.3 nM.
|Selective||CYP2C9, Ki: 19.3 nM|
Apigenin is a potent P450 inhibitor for CYP2C9 with Ki of 2 μM.
|Selective||CYP2C9, Ki: 2 μM|
Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.
Pioglitazone HCl is a hydrochloride salt form of pioglitazone which is a cytochrome P450 (CYP)2C8 and CYP3A4 enzymes inhibitor for CYP2C8, CYP3A4 and CYP2C9 with Ki of 1.7 μM, 11.8 μM and 32.1 μM, respectively.
|Pan||CYP2C9, Ki: 32.1 μM; CYP2C8, Ki: 1.7 μM|
Avasimibe inhibits ACAT with IC50 of 3.3 μM, also inhibits human P450 isoenzymes CYP2C9, CYP1A2 and CYP2C19 with IC50 of 2.9 μM, 13.9 μM and 26.5 μM, respectively.
|Pan||CYP2C19, IC50: 26.5 μM; CYP2C9, IC50: 2.9 μM|
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