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Norepinephrine

Other Neuronal Signaling Related Inhibitors

Secretase GluR GABA Receptor Dopamine Receptor 5-HT Receptor P2 Receptor AChR Histamine Receptor MAO Beta Amyloid
Cat.No. Product Name Information Product Use Citations Product Validations
S3199 Reboxetine mesylate Reboxetine (PNU 155950E) is a norepinephrine reuptake inhibitor with Ki of 8.2 nM.
Cancer Discov, 2020, CD-20-0160
Micromachines (Basel), 2018, 9(6)E274
S1444 Ziprasidone HCl Ziprasidone HCl (CP-88059) is a novel and potent dopamine and serotonin (5-HT) receptor antagonist, used in the treatment of schizophrenia and bipolar disorder.
Scientific Reports, August 17, 2017, 8491
UNIVERSITY OF PÉCS, 2023,
Anticancer Res, 2021, 41(2):687-697
Verified customer review of Ziprasidone HCl
S2541 Clomipramine HCl Clomipramine HCl is a tricyclic antidepressant acting as a potent inhibitor of 5-HT reuptake with an IC50 value of 1.5 nM. Clomipramine hydrochloride is used in research on depression, anxiety, and obsessive-compulsive disorder (OCD).
Infectious Medicine, 2024, 100130
Biomed Pharmacother, 2022, 153:113328
Pharmaceuticals, 2022, 241
S2084 Duloxetine HCl Duloxetine HCl (LY-248686) is a serotonin-norepinephrine reuptake inhibitor with Ki of 4.6 nM, used for treatment of major depressive disorder and generalized anxiety disorder (GAD).
Autophagy, 2026, 1-27.
Cancers (Basel), 2022, 14(19)4883
Drug Metab Dispos, 2015, 44(3):378-88
Verified customer review of Duloxetine HCl
S3183 Amitriptyline HCl Amitriptyline HCl is an inhibitor of both serotonin transporter (SERT) and norepinephrine transporter (NET) with Ki of 3.45 nM and 13.3 nM, respectively. This compound also inhibits histamine receptor H1, histamine receptor H4, 5-HT2 and sigma 1 receptor with Ki of 0.5 nM, 7.31 nM, 235 nM and 287 nM, respectively. It is a tricyclic antidepressant (TCA).
Proceedings of the National Academy of Sciences, 2021, e2026403118
Environ Toxicol Chem, 2021, 10.1002/etc.5018
PLoS Pathog, 2020, 16;16(3):e1008341
S2517 Maprotiline HCl Maprotiline HCl is a selective noradrenalin re-uptake inhibitor, used in the treatment of depression.
Annals of Hematology, September 2, 2025, 5841-5854
Annals of Hematology, September 02, 2025, 5841-5854
Frontiers in Pharmacology, May 20, 2021, 689767
S5947 Amitriptyline Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties, widely used to treat depression and neuropathic pain. This compound is an inhibitor of both serotonin transporter (SERT) and norepinephrine transporter (NET) with Ki of 3.45 nM and 13.3 nM, respectively. It also inhibits histamine receptor H1, histamine receptor H4, 5-HT2 and sigma 1 receptor with Ki of 0.5 nM, 7.31 nM, 235 nM and 287 nM, respectively. This product is a waxy solid.
Cancer Cell, 2025, 43(4):776-796.e14
Cancer Cell, 2025, 776-796.e14
Proceedings of the National Academy of Sciences, 2021, e2026403118
S3698 Nortriptyline hydrochloride Nortriptyline hydrochloride (Desitriptyline, ELF-101, EN-7048, Desmethylamitriptyline) is the hydrochloride salt form of nortriptyline, a tricyclic antidepressant agent used for short-term treatment of various forms of depression.
Frontiers in Bioinformatics, September 14, 2021, 710591
EMBO Molecular Medicine, December 23, 2025, 433-461
EMBO Molecular Medicine, December 23, 2025, Epub ahead of print
S2292 Diosmin Diosmin is an agonist of the aryl hydrocarbon receptor (AhR). This compound is a semisynthetic phlebotropic agent and a flavonoid found in a variety of citrus fruits.
The Indonesian Biomedical Journal, February 2024, 56-65
Int J Mol Sci, 2020, 21(14):5025
Mol Biol Rep, 2020, 47(3):2217-2230
S4113 Desvenlafaxine Desvenlafaxine (WY 45233 Succinate) is a serotonin (5-HT) and norepinephrine (NE) reuptake inhibitor with Ki of 40.2 nM and 558.4 nM, respectively.
Am J Cancer Res, 2024, 14(3):1087-1100
American Journal of Cancer Research, 2024, 1087-1100
Drug Metab Dispos, 2020, 48(10):1044-1052