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Cat.No. Product Name Information Product Use Citations Product Validations
S1346 Heparin sodium Heparin sodium, a sulfated polysaccharide belonging to the family of glycosaminoglycans, has numerous important biological activities associated with its interaction with diverse proteins. Heparin is used as an anticoagulant primarily through its interaction with AT III by enhancing AT-IIImediated inhibition of blood coagulation factors, including thrombin and factor Xa. Heparin prevents the induction of autophagy.
Cell Rep Med, 2025, 6(10):102410
Bone Res, 2025, 13(1):37
Theranostics, 2025, 15(6):2597-2623
S2196 Dabigatran Dabigatran is a potent nonpeptide thrombin inhibitor with an IC50 of 9.3 nM in a cell-free assay.
Thromb Res, 2025, 255:109480
Thromb Haemost, 2025, 10.1055/a-2497-4213
Thromb Haemost, 2024, 10.1055/a-2483-0107
Verified customer review of Dabigatran
S2154 Dabigatran (BIBR-1048) etexilate Dabigatran Etexilate (BIBR-1048) is the prodrug of dabigatran, a potent, nonpeptidic small molecule that specifically and reversibly inhibits both free and clot-bound thrombin by binding to the active site of the thrombin molecule.
J Immunother Cancer, 2024, 12(11)e009805
Eur J Pharmacol, 2024, 985:177058
Sci Rep, 2022, 12(1):3955
Verified customer review of Dabigatran (BIBR-1048) etexilate
S2069 Argatroban (MCI-9038) Argatroban (MCI-9038) is a potent and selective synthetic thrombin inhibitor, with Ki ranging from 5 nM to 39 nM, and it is used as an anticoagulant.
J Immunother Cancer, 2024, 12(11)e009805
Neural Regen Res, 2024, 19(2):434-439
Cancer Lett, 2023, 553:215983
S5074 Argatroban Monohydrate Argatroban (Argatroban hydrate, Argipidine,MCI-9038 Monohydrate) is a direct, selective thrombin inhibitor with anticoagulant effects.
Cancer Lett, 2023, 553:215983
Life Sci, 2021, 269:119073
S5960 Dabigatran etexilate mesylate Dabigatran etexilate mesylate (Pradaxa, BIBR 1048MS, Dabigatran etexilate methanesulfonate) is an orally active prodrug of Dabigatran which is a reversible and selective, direct thrombin inhibitor (DTI). Dabigatran selectively and reversibly inhibits human thrombin with Ki of 4.5 nM and thrombin-induced platelet aggregation with IC50 of 10 nM.
bioRxiv, 2020, 10.1101/2020.04.22.054981
E5835New Heparin Heparin is a highly sulfated polysaccharide primarily used as an anticoagulant, which works mainly by inhibiting thrombin (FIIa) and/or factor Xa (FXa). It is commonly used to prevent and treat thromboembolic conditions such as deep vein thrombosis and pulmonary embolism. It also plays roles in inflammation, angiogenesis, and growth factor signaling, with potential therapeutic applications in cancer treatment and allergic conditions.