| Cat.No. |
Product Name |
Information |
|
S7083
|
LDK378
|
LDK378 is an orally available ALK inhibitor with IC50 of 0.15 nM.
|
|
S7039
|
PD168393
|
|
|
S4911
|
BMS-690514
|
BMS-690514 is a potent inhibitor of EGFR and VEGFR2 with IC50 of 5 nM and 50 nM, respectively.
|
|
S8042
|
GW2580
|
GW2580 is a selective inhibitor of human c-FMS with IC50 of 30 nM.
|
|
S7067
|
EMD 1214063
|
EMD 1214063 is a potent and selective c-Met inhibitor with IC50 of 6 nM.
|
|
S4001
|
Cabozantinib malate
|
Cabozantinib malate is the malate of Cabozantinib, a potent VEGFR2 inhibitor with IC50 of 0.035 nM and also inhibits c-Met, Ret, Kit, Flt-1/3/4, Tie2, and AXL with IC50 of 1.3 nM, 4 nM, 4.6 nM, 12 nM/11.3 nM/6 nM, 14.3 nM and 7 nM, respectively.
|
|
S8024
|
Tyrphostin AG 1296 (AG 1296)
|
Tyrphostin AG 1296 (AG 1296) is an inhibitor of PDGFR, FGFR and c-Kit with IC50 of < 1 μM, 12.3 μM and 1.8 μM, respectively.
|
|
S7000
|
AP26113
|
AP26113 is a potent ALK inhibitor for ALK, FER, ROS/ROS1, FLT3 and FES/FPS with IC50 of 0.62 nM, 1.3 nM, 1.9 nM, 2.1 nM and 3.4 nM, respectively.
|
|
S8009
|
AG 18 (Tyrphostin 23)
|
AG 18 inhibits EGFR with IC50 of 35 μM.
|
|
S8003
|
PQ 401
|
PQ 401 is an IGF-1R inhibitor with IC50 of <1 μM.
|