• Inhibitory Selectivity
  • Solubility
Catalog No. Product Name Solubility(25°C)
Water DMSO Alcohol
S7928 DASA-58 <1 mg/mL 91 mg/mL <1 mg/mL
S8616 PKM2 inhibitor(compound 3k) <1 mg/mL 6 mg/mL <1 mg/mL
Catalog No. Information Product Use Citations Product Validations


DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator.


PKM2 inhibitor(compound 3k)

PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.

Tags: PKM activator | PKM inhibitor | PKM modulator |PKM activity