DREADD agonist 21

Catalog No.S0457

For research use only.

DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (hM3Dq) with EC50 of 1.7 nM.

DREADD agonist 21 Chemical Structure

CAS No. 56296-18-5

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Biological Activity

Description DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (hM3Dq) with EC50 of 1.7 nM.
Targets
hM3Dq [1]
(Cell-free assay)
1.7 nM(EC50)

Protocol (from reference)

Solubility (25°C)

In vitro

Chemical Information

Molecular Weight 278.35
Formula

C17H18N4

CAS No. 56296-18-5
Storage 3 years -20°C powder
2 years -80°C in solvent
Smiles C1CN(CCN1)C2=NC3=CC=CC=C3NC4=CC=CC=C42

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