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P450 Inhibitors

  • Cat.No
  • Product Name
  • Information
  • Publications
  • Customer Reviews
  • S1442
  • Voriconazole
  • Voriconazole (VFEND) is a triazole antifungal medication that is generally used to treat serious, invasive fungal infections.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2246
  • Abiraterone Acetate (CB7630)
  • Abiraterone Acetate (CB 7630) is a highly active and selective 17α-hydroxylase/17,20 lyase (CYP17A1) inhibitor with an IC50 of 72 nM.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2187
  • Avasimibe(CI-1011)
  • Avasimibe(CI-1011) is a novel orally bioavailable acyl coenzyme A:cholesterol acyltransferase inhibitor with IC50 of 2.9, 13.9, 26.5 μM for CYP2C9, CYP1A2, and CYP2C19
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2268
  • Baicalein
  • Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2401
  • Sodium Danshensu
  • Sodium Danshensu is a mono sodium of danshensu which is a compound isolated from Salvia miltiorrhiza Bge.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2757
  • TH-302
  • TH-302 is a selectively targeting hypoxic regions of solid tumors hypoxia-activated prodrug with an IC50 of 19 nM.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2394
  • Naringenin
  • Naringenin is a flavonoid that is considered to have a bioactive effect on human health as antioxidant, free radical scavenger, anti-inflammatory, carbohydrate metabolism promoter, and immune system modulator.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • S2262
  • Apigenin
  • Apigenin is a potent CYP2C9 inhibitor with an IC50 of 23 pM.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2136
  • Cytochrome P450 14a-demethylase inhibitor 1b
  • Cytochrome P450 14a-demethylase inhibitor 1b is an antifungal agent and an analog of fluconazole with an MIC80 of 3.9 ng/ml against Candida albicans and Microsporum gypseum.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2137
  • Cytochrome P450 14a-demethylase inhibitor 1c
  • Cytochrome P450 14a-demethylase inhibitor 1c is an antifungal agent and an analog of fluconazole with an MIC80 of 15.6 ng/ml against Candida albicans and Microsporum gypseum.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)
  • water-soluble S2138
  • Cytochrome P450 14a-demethylase inhibitor 1d
  • Cytochrome P450 14a-demethylase inhibitor 1d is an antifungal agent and an analog of fluconazole with an MIC80 of 15.6 ng/ml against Candida albicans and Microsporum gypseum.
  • 0 Reference(s) (0)
  • (0)Review(s) (0)